SCHEMBL5205702

SCHEMBL5205702

C=CCn1cc(C2CCN(C(=O)c3ccc(C)c(C(=O)c4ccc(C)cc4C=CC)c3)C2)c2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 6/20 0.37
CNR2 P34972 1/20 0.37
HSD11B1 P28845 3/20 0.36
HRH2 P25021 2/20 0.36
USP2 O75604 1/20 0.35
FASN P49327 1/20 0.34
MYC P01106 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5201910 0.81 NPC1 (0.42) CNR1CNR2HRH2MAPTHTT
SCHEMBL4860169 0.72 MAPT (0.40) HRH2MAPT
SCHEMBL4860164 0.70 CNR2 (0.36) CNR2HRH2MAPT
SCHEMBL5203731 0.69 PDE2A (0.41) CNR1HSD11B1
SCHEMBL5202510 0.69 HSD11B1 (0.55) CNR1HSD11B1HRH2HTT
SCHEMBL4858356 0.68 CREBBP (0.42) CNR1HSD11B1HRH2
SCHEMBL4862667 0.68 TSHR (0.47) CNR2HSD11B1HRH2
SCHEMBL5205358 0.68 ALDH1A1 (0.45) HSD11B1HRH2
SCHEMBL5201671 0.67 ALDH1A1 (0.51) CNR1CNR2HRH2MAPTHTT
SCHEMBL6378962 0.67 HRH2 (0.34) CNR2HRH2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP disclosed