SCHEMBL4860169

SCHEMBL4860169

C=CCn1cc(C2CCN([C](C=Cc3ccc(C)cc3)C(=O)c3ccc(C)cc3)C2)c2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.40
KDM4E B2RXH2 2/20 0.40
LMNA P02545 2/20 0.40
TP53 P04637 2/20 0.40
THRB P10828 1/20 0.40
NPC1 O15118 3/20 0.39
HPGD P15428 3/20 0.39
RAB9A P51151 3/20 0.39
ALDH1A1 P00352 3/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
CCR2 P41597 2/20 0.38
HDAC1 Q13547 3/20 0.38
HDAC3 O15379 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5201910 0.85 NPC1 (0.42) MAPTLMNANPC1RAB9AMEN1
SCHEMBL4858356 0.77 CREBBP (0.42) ALDH1A1HDAC1HDAC3HDAC2HDAC10
SCHEMBL4860164 0.73 CNR2 (0.36) MAPTKDM4ELMNATP53NPC1
SCHEMBL5205702 0.72 CNR1 (0.37) MAPTHRH2
SCHEMBL5203731 0.71 PDE2A (0.41) ALDH1A1SMN1; SMN2
SCHEMBL6378962 0.70 HRH2 (0.34) MAPTKDM4ELMNATP53NPC1
SCHEMBL5206944 0.70 RAB9A (0.55) MAPTKDM4ELMNANPC1HPGD
SCHEMBL4858050 0.68 RAB9A (0.62) MAPTKDM4ELMNATP53THRB
SCHEMBL5202510 0.68 HSD11B1 (0.55) ALDH1A1KMT2ASMN1; SMN2HRH2
SCHEMBL5202293 0.67 THRB (0.49) MAPTKDM4ELMNATHRBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7368470-B2 Substituted 3-pyrrolidine-indole derivatives GRUENENTHAL GMBH (DE) 2008-05-06 US disclosed