SCHEMBL5206469

SCHEMBL5206469

COc1ccc(C(C)N2CCN(C(=O)c3cccnc3)CC2CC(N)=O)cc1OC

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.50
TDP1 Q9NUW8 1/20 0.46
CSF1R P07333 1/20 0.45
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 1/20 0.45
KLK7 P49862 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43
PDGFRB P09619 1/20 0.42
SLC18A3 Q16572 1/20 0.40
MMP1 P03956 1/20 0.40
MMP3 P08254 1/20 0.40
MMP7 P09237 1/20 0.40
MMP9 P14780 1/20 0.40
MMP13 P45452 1/20 0.40
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5206464 0.80 POLB (0.51) POLBTDP1CSF1RALDH1A1KDM4E
SCHEMBL5192047 0.80 KMT2A (0.45) TDP1ALDH1A1GAA
SCHEMBL5193931 0.78 HIF1A (0.42) ALDH1A1
SCHEMBL5213600 0.76 ALDH1A1 (0.51) POLBALDH1A1
SCHEMBL5193553 0.73 PDGFRB (0.45) PDGFRB
SCHEMBL5206448 0.73 POLB (0.45) POLBTDP1CSF1RALDH1A1KDM4E
SCHEMBL5192328 0.73 TDP1 (0.52) POLBTDP1ALDH1A1KDM4EKLK7
SCHEMBL5191190 0.73 HIF1A (0.47) POLBALDH1A1
SCHEMBL5189720 0.71 NOS2 (0.54)
SCHEMBL27402749 0.71 SMN1; SMN2 (0.46) POLBALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP disclosed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP disclosed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO disclosed