SCHEMBL5192047

SCHEMBL5192047

CC(c1cccs1)N1CCN(C(=O)c2cccnc2)CC1CC(N)=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.45
ALDH1A1 P00352 2/20 0.43
MAPK1 P28482 2/20 0.43
CYP2C19 P33261 1/20 0.43
CTSL P07711 1/20 0.41
CTSB P07858 1/20 0.41
CASP3 P42574 1/20 0.41
CTSK P43235 1/20 0.41
CTSF Q9UBX1 1/20 0.41
TDP1 Q9NUW8 1/20 0.39
FABP6 P51161 1/20 0.39
GAA P10253 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA7 P36544 1/20 0.39
CHRNA4 P43681 1/20 0.39
VNN1 O95497 1/20 0.39
PKM P14618 1/20 0.39
PIK3CD O00329 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5206469 0.80 POLB (0.50) ALDH1A1TDP1GAA
SCHEMBL5191020 0.75 SMN1; SMN2 (0.43) KMT2ACYP2C19
SCHEMBL5193832 0.72 FABP6 (0.46) KMT2AALDH1A1MAPK1TDP1FABP6
SCHEMBL27402749 0.71 SMN1; SMN2 (0.46) KMT2AALDH1A1MAPK1FABP6CHRNB2
SCHEMBL5192328 0.70 TDP1 (0.52) KMT2AALDH1A1TDP1
SCHEMBL27401275 0.70 ALDH1A1 (0.44) KMT2AALDH1A1FABP6CHRNB2CHRNB4
SCHEMBL5281219 0.69 ALDH1A1 (0.49) KMT2AALDH1A1MAPK1CYP2C19CTSL
SCHEMBL27411591 0.69 FABP6 (0.47) KMT2AALDH1A1MAPK1TDP1FABP6
SCHEMBL5206464 0.68 POLB (0.51) ALDH1A1MAPK1TDP1
SCHEMBL5190965 0.68 CHRNB2 (0.51) KMT2AALDH1A1MAPK1GAACHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP claimed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP claimed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO claimed