SCHEMBL5207531

SCHEMBL5207531

Cc1cnc(Cl)nc1Cc1cccc(C(F)(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
HSP90AA1 P07900 1/20 0.44
P2RX3 P56373 1/20 0.43
HTR2C P28335 2/20 0.42
HTR2B P41595 2/20 0.42
GPR52 Q9Y2T5 3/20 0.41
HTR2A P28223 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
LTA4H P09960 1/20 0.40
SCN8A Q9UQD0 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5203839 0.81 CYP1A2 (0.46) RAB9ACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL15504928 0.80 YTHDC1 (0.41) TAAR1
SCHEMBL27955757 0.78 PIN1 (0.38) HSP90AA1TAAR1
SCHEMBL5209985 0.76 HSP90AA1 (0.39) RAB9ACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL28227779 0.72 CYP1A2 (0.46) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL8871754 0.71 GPR52 (0.42) RAB9ACYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL3237564 0.71 TAAR1 (0.64) HTR2CHTR2BHTR2ALTA4HTAAR1
SCHEMBL9492711 0.70 HTR2C (0.48) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL31414537 0.69 LMNA (0.59) CYP1A2CYP3A4CYP2D6CYP2C19HSP90AA1
SCHEMBL857569 0.69 HTR2A (0.42) RAB9AHSP90AA1HTR2CHTR2BGPR52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1036066-B1 SUBSTITUTED PYRIMIDINE AND PYRIDINE HERBICIDES MID AMERICA COMMERCIALIZATION (US) 2007-04-18 EP disclosed
US-20040033896-A1 E.g., 5-ethyl-4-((3 -(trifluoromethoxy)phenyl)methyl)-2-(3-(trifluoromethyl)-1H pyrazol-1-yl)pyrimidine and 5-methyl-2-(4-(trifluoromethyl)phenyl)-4-((3-(trifluoromethyl) phenyl)methyl)pyrimidine KOETHER GERARD (US) 2004-02-19 US disclosed
US-6525001-B1 5-methyl-2-(4-(trifluoromethyl)phenyl)-4-((3 -(trifluoromethyl)phenyl)methyl)pyrimidine MID-AMERICAN COMMERCIALIZATION CORPORATION 2003-02-25 US disclosed
EP-1036066-A1 SUBSTITUTED PYRIMIDINE AND PYRIDINE HERBICIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 2000-09-20 EP disclosed
WO-1999028301-A1 SUBSTITUTED PYRIMIDINE AND PYRIDINE HERBICIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1999-06-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040033896-A1 E.g., 5-ethyl-4-((3 -(trifluoromethoxy)phenyl)methyl)-2-(3-(trifluoromethyl)-1H pyrazol-1-yl)pyrimidine and 5-methyl-2-(4-(trifluoromethyl)phenyl)-4-((3-(trifluoromethyl) phenyl)methyl)pyrimidine PYM1, Q6ZSR9, MRM1 RAB9A 1261/4885CYP1A2 429/4885CYP3A4 724/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.