SCHEMBL5209607

SCHEMBL5209607

Cc1cc(-c2c(Cl)ccc(C(=O)O)c2Cl)on1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
TSHR P16473 3/20 0.54
KDM4E B2RXH2 1/20 0.54
USP2 O75604 1/20 0.54
HCAR2 Q8TDS4 1/20 0.42
RARA P10276 1/20 0.40
RARB P10826 1/20 0.40
RARG P13631 1/20 0.40
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
MAPK1 P28482 1/20 0.39
CSF1R P07333 5/20 0.39
PRKAG1 P54619 1/20 0.38
PRKAA1 Q13131 1/20 0.38
PRKAB1 Q9Y478 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NTRK1 P04629 1/20 0.38
TP53 P04637 1/20 0.37
CASP1 P29466 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5204512 0.89 KDM4E (0.43) ALDH1A1TSHRKDM4EUSP2HCAR2
SCHEMBL8137248 0.85 NOTUM (0.47) ALDH1A1TSHRKDM4EUSP2KMT2A
SCHEMBL8138255 0.84 ALDH1A1 (0.49) ALDH1A1TSHRKDM4EUSP2HCAR2
SCHEMBL8135897 0.83 ALDH1A1 (0.48) ALDH1A1TSHRKDM4EUSP2HCAR2
SCHEMBL7988196 0.80 KDM4E (0.50) ALDH1A1TSHRKDM4EUSP2HCAR2
SCHEMBL5204516 0.77 ALDH1A1 (0.35) ALDH1A1TSHRKDM4EUSP2KMT2A
SCHEMBL27513006 0.77 ALDH1A1 (0.74) ALDH1A1TSHRKDM4EUSP2HCAR2
SCHEMBL8377155 0.76 NTRK1 (0.35) ALDH1A1TSHRKDM4EUSP2KMT2A
SCHEMBL8306233 0.75 SMN1; SMN2 (0.39) ALDH1A1TSHRKDM4EUSP2KMT2A
SCHEMBL8522694 0.75 ALDH1A1 (0.42) ALDH1A1TSHRKDM4ERARARARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5948917-A INTERMEDIATE FOR THE PRODUCTION OF A HERBICIDALLY ACTIVE PYRAZOLE COMPOUND NIPPON SODA CO., LTD. (JP) 1999-09-07 US claimed
EP-0891972-A1 3-(ISOXAZOL-5-YL)-SUBSTITUTED BENZOIC ACID DERIVATIVES AND PROCESS FOR PRODUCING THE SAME NIPPON SODA CO., LTD. (JP) 1999-01-20 EP claimed
EP-0958292-B1 4-(3-HETEROCYCLYL-1-BENZOYL)PYRAZOLES AND THEIR USE AS HERBICIDES BASF AG (DE) 2007-01-03 EP disclosed
US-6165944-A 4-(3-heterocyclyl-1-benzoyl) pyrazoles and their use as herbicides BASF AKTIENGESELLSCHAFT (DE) 2000-12-26 US disclosed
US-6100421-A METHYL 3-FORMYL-4-METHANESULFONYL-2-METHYLBENZOATE, USEFUL AS A STARTING MATERIAL FOR HERBICIDE MANUFACTURE NIPPON SODA CO., LTD. (JP) 2000-08-08 US disclosed
US-5948917-A INTERMEDIATE FOR THE PRODUCTION OF A HERBICIDALLY ACTIVE PYRAZOLE COMPOUND NIPPON SODA CO., LTD. (JP) 1999-09-07 US disclosed
EP-0894792-A1 HETEROCYCLE-SUBSTITUTED BENZENE DERIVATIVES AND HERBICIDES NIPPON SODA CO., LTD. (JP) 1999-02-03 EP disclosed
EP-0891972-A1 3-(ISOXAZOL-5-YL)-SUBSTITUTED BENZOIC ACID DERIVATIVES AND PROCESS FOR PRODUCING THE SAME NIPPON SODA CO., LTD. (JP) 1999-01-20 EP disclosed