SCHEMBL5211458

SCHEMBL5211458

CCSc1nc(N)cc(-c2ccccc2-c2ccc(OC)c(Cl)c2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.46
PTGS1 P23219 1/20 0.46
ADORA2A P29274 2/20 0.46
ADORA1 P30542 2/20 0.46
MAPK1 P28482 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.42
AGPAT2 O15120 4/20 0.39
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
GAA P10253 1/20 0.38
HRH4 Q9H3N8 1/20 0.37
DCK P27707 1/20 0.37
PGK1 P00558 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
TP53 P04637 1/20 0.36
TSHR P16473 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6504950 0.78 KDM4E (0.48) MAPK1SMN1; SMN2DCKMEN1KMT2A
SCHEMBL5181345 0.74 ADORA1 (0.51) PTGS2PTGS1ADORA2AADORA1MAPK1
SCHEMBL5305206 0.73 PTGS2 (0.53) PTGS2PTGS1ADORA2AADORA1SMN1; SMN2
SCHEMBL3602925 0.72 HSP90AA1 (0.51) MAPK1SMN1; SMN2HSP90AA1HSP90AB1MEN1
SCHEMBL5277858 0.69 HRH4 (0.48) PTGS2PTGS1ADORA2AADORA1HSP90AA1
SCHEMBL3450830 0.69 TUBB4A (0.49) MAPK1AGPAT2GAAMEN1KMT2A
SCHEMBL5191007 0.69 RAB9A (0.48) ADORA2AADORA1SMN1; SMN2HSP90AA1GAA
SCHEMBL25129319 0.68 PTGS2 (0.63) PTGS2PTGS1ADORA2AADORA1
SCHEMBL31074324 0.68 PTGS2 (0.63) PTGS2PTGS1ADORA2AADORA1
SCHEMBL28811659 0.67 MCHR1 (0.56) PTGS2PTGS1ADORA2AADORA1HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1796673-A2 NOVEL PYRIMIDINE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM Reddy US Therapeutics, Inc. (US) 2007-06-20 EP disclosed
WO-2006034473-A2 NOVEL PYRIMIDINE COMPOUNDS, PROCESS FOR THEIR PREPARATION AND COMPOSITIONS CONTAINING THEM REDDY US THERAPEUTICS, INC. (US) 2006-03-30 WO disclosed