SCHEMBL5215152

SCHEMBL5215152

O=C(Nc1ccccc1)Sc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
EPHX2 P34913 2/20 0.54
EPHX1 P07099 1/20 0.54
TSHR P16473 1/20 0.54
CDK9 P50750 1/20 0.54
CLK4 Q9HAZ1 1/20 0.54
HSD17B10 Q99714 2/20 0.50
NAPRT Q6XQN6 1/20 0.50
POLB P06746 2/20 0.49
MAPT P10636 2/20 0.49
KMT2A Q03164 2/20 0.49
MEN1 O00255 1/20 0.49
MAPK1 P28482 1/20 0.49
ALDH1A1 P00352 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
IDO1 P14902 1/20 0.47
CASP3 P42574 1/20 0.47
SENP7 Q9BQF6 1/20 0.47
MAOA P21397 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14599306 0.88 MAOA (0.58) TP53SMN1; SMN2EPHX2EPHX1TSHR
SCHEMBL27568887 0.87 SMN1; SMN2 (0.51) TP53SMN1; SMN2EPHX2EPHX1TSHR
SCHEMBL22648045 0.87 NPC1 (0.56) TP53SMN1; SMN2HSD17B10POLBMAPT
SCHEMBL8616935 0.85 KMT2A (0.61) SMN1; SMN2POLBMAPTKMT2AMEN1
SCHEMBL22648006 0.82 CRHBP (0.52) TP53SMN1; SMN2POLBMAPTKMT2A
SCHEMBL22648796 0.82 RAB9A (0.52) TP53SMN1; SMN2EPHX1TSHRPOLB
SCHEMBL11869490 0.82 HSD17B10 (0.56) TP53SMN1; SMN2TSHRHSD17B10NAPRT
SCHEMBL12132227 0.79 EPHX2 (0.61) TP53SMN1; SMN2EPHX2EPHX1TSHR
SCHEMBL3067346 0.79 EPHX2 (0.61) TP53SMN1; SMN2EPHX2EPHX1TSHR
SCHEMBL11285224 0.79 MAPT (0.49) TP53SMN1; SMN2EPHX2EPHX1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11046645-B2 Isothiocyanate production method, composition for transporting and storing N-substituted O-substituted thiocarbamate, and isothiocyanate composition ASAHI KASEI CHEMICALS CORPORATION (JP) 2021-06-29 US disclosed
EP-3363785-B1 ISOTHIOCYANATE PRODUCTION METHODS ASAHI CHEMICAL IND (JP) 2020-09-16 EP disclosed
US-20190233371-A1 Isothiocyanate Production Method, Composition for Transporting and Storing N-Substituted O-Substituted Thiocarbamate, and Isothiocyanate Composition ASAHI KASEI KABUSHIKI KAISHA (JP) 2019-08-01 US disclosed
EP-3214071-B1 ISOTHIOCYANATE COMPOSITION ASAHI CHEMICAL IND (JP) 2019-07-03 EP disclosed
US-10308601-B2 Isothiocyanate production method, composition for transporting and storing N-substituted O-substituted thiocarbamate, and isothiocyanate composition ASAHI KASEI CHEMICALS CORPORATION (JP) 2019-06-04 US disclosed
EP-3363785-A1 ISOTHIOCYANATE PRODUCTION METHODS Asahi Kasei Chemicals Corporation (JP) 2018-08-22 EP disclosed
EP-3214071-A1 ISOTHIOCYANATE COMPOSITION Asahi Kasei Chemicals Corporation (JP) 2017-09-06 EP disclosed
US-20160016901-A1 ISOTHIOCYANATE PRODUCTION METHOD, COMPOSITION FOR TRANSPORTING AND STORING N-SUBSTITUTED O-SUBSTITUTED THIOCARBAMATE, AND ISOTHIOCYANATE COMPOSITION ASAHI KASEI CHEMICALS CORPORATION (JP) 2016-01-21 US disclosed
EP-2966060-A1 ISOTHIOCYANATE PRODUCTION METHOD, COMPOSITION FOR TRANSPORTING AND STORING N-SUBSTITUTED O-SUBSTITUTED THIOCARBAMATE, AND ISOTHIOCYANATE COMPOSITION Asahi Kasei Chemicals Corporation (JP) 2016-01-13 EP disclosed
EP-1660469-B1 PROCESS FOR THE PREPARATION OF 11-(1-PIPERAZINYL)DIBENZO 'B, F! '1 ,4!-THIAZEPINE, AN INTERMEDIATE IN THE SYNTHESIS OF THE ANTIPSYCHOTIC DRUG QUETIAPINE HELM AG (DE) 2007-08-29 EP disclosed
EP-1660469-A1 PROCESS FOR THE PREPARATION OF 11-(1-PIPERAZINYL)DIBENZO 'B, F! '1 ,4!-THIAZEPINE, AN INTERMEDIATE IN THE SYNTHESIS OF THE ANTIPSYCHOTIC DRUG QUETIAPINE Helm AG (DE) 2006-05-31 EP disclosed
WO-2005012274-A1 PROCESS FOR THE PREPARATION OF 11-(1-PIPERAZINYL)DIBENZO `B, F! `1 ,4!-THIAZEPINE, AN INTERMEDIATE IN THE SYNTHESIS OF THE ANTIPSYCHOTIC DRUG QUETIAPINE HELM AG (DE) 2005-02-10 WO disclosed
US-4835312-A Production process of N-substituted amide compounds MITSUI CHEMICALS, INCORPORATED (JP) 1989-05-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11046645-B2 Isothiocyanate production method, composition for transporting and storing N-substituted O-substituted thiocarbamate, and isothiocyanate composition TST, SLCO4C1, SLCO2B1 TP53 3955/4885SMN1; SMN2 4351/4885EPHX2 1370/4885
US-20160016901-A1 ISOTHIOCYANATE PRODUCTION METHOD, COMPOSITION FOR TRANSPORTING AND STORING N-SUBSTITUTED O-SUBSTITUTED THIOCARBAMATE, AND ISOTHIOCYANATE COMPOSITION TST, SLCO4C1, SLCO2B1 TP53 3955/4885SMN1; SMN2 4351/4885EPHX2 1370/4885
US-20190233371-A1 Isothiocyanate Production Method, Composition for Transporting and Storing N-Substituted O-Substituted Thiocarbamate, and Isothiocyanate Composition TST, SLCO4C1, SLCO2B1 TP53 3955/4885SMN1; SMN2 4351/4885EPHX2 1370/4885
US-10308601-B2 Isothiocyanate production method, composition for transporting and storing N-substituted O-substituted thiocarbamate, and isothiocyanate composition TST, SLCO4C1, SLCO2B1 TP53 3955/4885SMN1; SMN2 4351/4885EPHX2 1370/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.