SCHEMBL5216286

SCHEMBL5216286

O=C(Cl)c1ccc(F)cc1I

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CES2 O00748 5/20 0.47
CES1 P23141 5/20 0.47
ALOX15 P16050 2/20 0.42
ALDH1A1 P00352 1/20 0.42
KEAP1 Q14145 1/20 0.38
TTR P02766 1/20 0.38
HPGD P15428 1/20 0.38
MAOB P27338 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
TAS1R2 Q8TE23 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
P2RX7 Q99572 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28423060 0.83 CES2 (0.47) CES2CES1ALOX15ALDH1A1KEAP1
SCHEMBL27883251 0.83 CES2 (0.50) CES2CES1ALDH1A1KEAP1TTR
SCHEMBL1588995 0.81 KEAP1 (0.53) CES2CES1ALDH1A1KEAP1TTR
SCHEMBL9834572 0.80 CES2 (0.52) CES2CES1ALOX15ALDH1A1KEAP1
SCHEMBL24006621 0.79 CES2 (0.47) CES2CES1ALDH1A1KEAP1TTR
SCHEMBL24013508 0.79 ALDH1A1 (0.46) CES2CES1ALDH1A1KEAP1HPGD
SCHEMBL165619 0.78 CES2 (0.68) CES2CES1ALOX15ALDH1A1KEAP1
SCHEMBL4727563 0.77 TPMT (0.37) CES2CES1ALOX15ALDH1A1
SCHEMBL23242477 0.77 CES2 (0.45) CES2ALOX15ALDH1A1KEAP1HPGD
SCHEMBL1626671 0.77 SMN1; SMN2 (0.47) ALDH1A1MAOBNPC1RAB9AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114835622-A N-tert-butyl protection-3-substituted indole compound and preparation method thereof 常州大学 2022-08-02 CN disclosed
CN-103848829-B Heteroaryl alkyne compounds and application thereof 南京圣和药业股份有限公司 2017-04-12 CN disclosed
CN-103848829-A Heteroaryl alkyne compounds and application thereof NANJING SANHOME PHARMACEUTICAL CO LTD 2014-06-11 CN disclosed
EP-1153013-B1 5-HT1F AGONISTS LILLY CO ELI (US) 2007-10-31 EP disclosed
US-6777428-B1 INHIBIT PEPTIDE EXTRAVASATION DUE TO STIMULATION OF THE TRIGEMINAL GANGLIA, AND ARE THEREFORE USEFUL FOR THE TREATMENT OF MIGRAINE AND ASSOCIATED DISORDERS ELI LILLY AND COMPANY 2004-08-17 US disclosed
CN-1149195-C 5-HTIF agonists 2004-05-12 CN disclosed
CN-1340045-A 5-HTIF agonists LILLY CO ELI (US) 2002-03-13 CN disclosed
EP-1153013-A2 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 2001-11-14 EP disclosed
WO-2000047559-A2 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 2000-08-17 WO disclosed