SCHEMBL9834572

SCHEMBL9834572

O=C(Cl)c1ccc(F)cc1C(=O)Cl

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CES2 O00748 7/20 0.52
CES1 P23141 7/20 0.52
KEAP1 Q14145 1/20 0.47
ALDH1A1 P00352 1/20 0.46
ALOX15 P16050 1/20 0.46
HPGD P15428 1/20 0.41
MAOB P27338 2/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
CA3 P07451 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CA5B Q9Y2D0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28516694 0.89 KEAP1 (0.57) CES2CES1KEAP1ALDH1A1ALOX15
SCHEMBL343535 0.84 CES2 (0.68) CES2CES1KEAP1ALDH1A1ALOX15
SCHEMBL165619 0.84 CES2 (0.68) CES2CES1KEAP1ALDH1A1ALOX15
SCHEMBL11588418 0.82 MAOB (0.49) CES2CES1KEAP1ALDH1A1ALOX15
SCHEMBL477556 0.82 CES2 (0.48) CES2CES1KEAP1ALDH1A1ALOX15
SCHEMBL5459423 0.82 MAOB (0.50) CES2CES1KEAP1ALDH1A1ALOX15
SCHEMBL106341 0.82 HPGD (0.54) CES2CES1ALDH1A1ALOX15HPGD
SCHEMBL1364589 0.80 CES2 (0.47) CES2CES1KEAP1ALDH1A1ALOX15
SCHEMBL4649267 0.80 CES2 (0.47) CES2CES1KEAP1ALDH1A1ALOX15
SCHEMBL31315010 0.80 CES2 (0.47) CES2CES1KEAP1ALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170255100-A1 DRY FILM STRUCTURE FUJIFILM ELECTRONIC MATERIALS U.S.A., INC. 2017-09-07 US disclosed
EP-0253837-B1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING BRANCHED ALKYL PYRIDINIUM SALTS MALLINCKRODT SPECIALTY CHEMICALS COMPANY (US) 1991-10-09 EP disclosed
EP-0252964-B1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING SUBSTITUTED PYRIDINIUM SALTS MALLINCKRODT SPECIALTY CHEMICALS COMPANY (US) 1991-08-21 EP disclosed
EP-0253838-B1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING N-SEC-ALKYL PYRIDINIUM SALTS MALLINCKRODT SPECIALTY CHEMICALS COMPANY (US) 1991-08-21 EP disclosed
US-4973771-A Phase transfer catalysts MALLINCKRODT, INC. (US) 1990-11-27 US disclosed
US-4973772-A Catalytic method for producing fluoroarmatic compounds using substituted pyridinium salts MALLINCKRODT, INC. (US) 1990-11-27 US disclosed
EP-0253836-B1 PREPARATION OF FLUOROAROMATIC COMPOUNDS IN DISPERSION OF POTASSIUM FLUORIDE Mallinckrodt, Inc. (a Delaware corporation) (US) 1990-10-03 EP disclosed
US-4927980-A REACTING CHLOROAROMATIC COMPOUND WITH ALKALI METAL FLUORIDE SALTS MALLINCKRODT INC. (US) 1990-05-22 US disclosed
US-4849552-A METHANOL, AROMATIC HYDROCARBON OR HALOCARBON, AZEOTROPES MALLINCKRODT, INC. (US) 1989-07-18 US disclosed
EP-0252964-A4 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING SUBSTITUTED PYRIDINIUM SALTS. MALLINCKRODT INC (US) 1988-07-14 EP disclosed
EP-0253836-A4 PREPARATION OF FLUOROAROMATIC COMPOUNDS IN DISPERSION OF POTASSIUM FLUORIDE. MALLINCKRODT INC (US) 1988-04-27 EP disclosed
EP-0253837-A4 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING BRANCHED ALKYL PYRIDINIUM SALTS. MALLINCKRODT INC (US) 1988-04-26 EP disclosed
EP-0253836-A1 PREPARATION OF FLUOROAROMATIC COMPOUNDS IN DISPERSION OF POTASSIUM FLUORIDE. MALLINCKRODT INC (US) 1988-01-27 EP disclosed
EP-0253837-A1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING BRANCHED ALKYL PYRIDINIUM SALTS. MALLINCKRODT INC (US) 1988-01-27 EP disclosed
EP-0252964-A1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING SUBSTITUTED PYRIDINIUM SALTS. MALLINCKRODT INC (US) 1988-01-20 EP disclosed
WO-1987004148-A1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING BRANCHED ALKYL PYRIDINIUM SALTS MALLINCKRODT, INC. (US) 1987-07-16 WO disclosed
WO-1987004151-A1 PREPARATION OF FLUOROAROMATIC COMPOUNDS IN DISPERSION OF POTASSIUM FLUORIDE MALLINCKRODT, INC. (US) 1987-07-16 WO disclosed
WO-1987004149-A1 PHASE TRANSFER CATALYSTS MALLINCKRODT, INC. (US) 1987-07-16 WO disclosed
WO-1987004150-A1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING SUBSTITUTED PYRIDINIUM SALTS MALLINCKRODT, INC. (US) 1987-07-16 WO disclosed