SCHEMBL5219484

SCHEMBL5219484

CCNc1cc(C(=O)O)cc(N2CCCCS2(O)O)c1C

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 12/20 0.44
BACE2 Q9Y5Z0 12/20 0.44
CTSD P07339 11/20 0.44
POLB P06746 1/20 0.38
GAA P10253 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
GFER P55789 1/20 0.36
PLEC Q15149 1/20 0.36
HCAR3 P49019 2/20 0.36
GPR35 Q9HC97 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
RPS6KB1 P23443 1/20 0.31
AKT1 P31749 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5219833 0.96 BACE1 (0.41) BACE1BACE2CTSDPOLBGAA
SCHEMBL5219490 0.89 BACE1 (0.50) BACE1BACE2CTSDPOLBGAA
SCHEMBL5218025 0.89 BACE1 (0.41) BACE1BACE2CTSDPOLBGAA
SCHEMBL5219825 0.86 BACE1 (0.47) BACE1BACE2CTSDPOLBGAA
SCHEMBL5220759 0.85 BACE1 (0.45) BACE1BACE2CTSDPOLBGAA
SCHEMBL5219381 0.84 GPR35 (0.37) BACE1BACE2CTSDPOLBGAA
SCHEMBL5218045 0.82 CTSD (0.42) BACE1BACE2CTSDGAAKDM4E
SCHEMBL5224401 0.79 POLB (0.35) POLBHTTHCAR3
SCHEMBL5218030 0.78 BACE1 (0.47) BACE1BACE2CTSDPOLBGAA
SCHEMBL5218055 0.76 CTSD (0.44) BACE1BACE2CTSDGAAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed