SCHEMBL5223624

SCHEMBL5223624

CCN1CCN(Cc2cnn(-c3ccc(-c4ccc(F)cc4)cc3)c2-c2c(C)noc2C)CC1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMO Q99835 5/20 0.41
PIK3CD O00329 1/20 0.39
MAPT P10636 3/20 0.38
DRD2 P14416 3/20 0.36
DRD4 P21917 3/20 0.36
DRD3 P35462 3/20 0.36
BRD4 O60885 4/20 0.35
LMNA P02545 2/20 0.35
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35
CYP1A2 P05177 1/20 0.35
ALOX15 P16050 1/20 0.35
APEX1 P27695 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35
HSD17B10 Q99714 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
GPR55 Q9Y2T6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224153 0.92 BRD4 (0.44) SMOPIK3CDMAPTDRD2DRD4
SCHEMBL5228017 0.89 SMO (0.39) SMOPIK3CDMAPTDRD2DRD4
SCHEMBL5225729 0.85 F10 (0.38) SMOPIK3CD
SCHEMBL5225124 0.83 PIK3CD (0.42) PIK3CDBRD4LMNAALDH1A1MEN1
SCHEMBL1998311 0.80 SMO (0.60) SMOMAPTDRD2DRD4DRD3
SCHEMBL5224916 0.79 SMO (0.44) SMOMAPTDRD2DRD4DRD3
SCHEMBL2761237 0.78 SMO (0.43) SMOMAPTDRD2DRD4DRD3
Hydrochloric Acid SCHEMBL1997589 0.77 SMO (0.42) SMOMAPTDRD2DRD4DRD3
SCHEMBL5227445 0.75 DRD4 (0.46) SMOMAPTDRD2DRD4DRD3
SCHEMBL5228219 0.74 SMO (0.47) SMOMAPTDRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed