SCHEMBL5228017

SCHEMBL5228017

Cc1noc(C)c1-c1c(CN2CCNCC2)cnn1-c1ccc(-c2ccc(F)cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 2/20 0.39
PIK3CD O00329 1/20 0.38
BRD4 O60885 7/20 0.38
BRD2 P25440 3/20 0.38
BRD3 Q15059 3/20 0.38
MAPT P10636 2/20 0.37
NPSR1 Q6W5P4 1/20 0.36
RIPK3 Q9Y572 1/20 0.36
CYP1A2 P05177 3/20 0.36
HSD17B10 Q99714 1/20 0.36
CYP3A4 P08684 1/20 0.36
HIF1A Q16665 1/20 0.36
LMNA P02545 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALDH1A1 P00352 1/20 0.34
GPR55 Q9Y2T6 1/20 0.34
ROCK2 O75116 1/20 0.34
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34
DRD3 P35462 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5223624 0.89 SMO (0.41) SMOPIK3CDBRD4MAPTCYP1A2
SCHEMBL5224153 0.89 BRD4 (0.44) SMOPIK3CDBRD4MAPTCYP1A2
SCHEMBL5225729 0.84 F10 (0.38) SMOPIK3CDROCK2
SCHEMBL5225124 0.80 PIK3CD (0.42) PIK3CDBRD4CYP1A2HSD17B10CYP3A4
SCHEMBL5228219 0.72 SMO (0.47) SMOMAPTLMNAL3MBTL1ALDH1A1
SCHEMBL5224744 0.70 HTR1A (0.38) SMOLMNAALDH1A1ROCK2
SCHEMBL5224916 0.69 SMO (0.44) SMOMAPTNPSR1LMNAL3MBTL1
SCHEMBL5227096 0.69 SMO (0.44) SMOMAPTNPSR1LMNAL3MBTL1
SCHEMBL5228124 0.68 SMO (0.43) SMOMAPTLMNAL3MBTL1DRD2
SCHEMBL5227160 0.68 SMO (0.41) SMOMAPTCYP1A2CYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed