SCHEMBL5225124

SCHEMBL5225124

Cc1noc(C)c1-c1c(CN(C)C)cnn1-c1ccc(-c2ccc(F)cc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.42
GPR55 Q9Y2T6 1/20 0.38
LMNA P02545 4/20 0.36
CYP1A2 P05177 4/20 0.36
CYP2C19 P33261 3/20 0.36
USP2 O75604 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
ALOX15 P16050 1/20 0.36
APEX1 P27695 1/20 0.36
KMT2A Q03164 1/20 0.36
HSD17B10 Q99714 1/20 0.36
PTGS2 P35354 1/20 0.35
BRD4 O60885 6/20 0.34
CYP3A4 P08684 2/20 0.34
TP53 P04637 1/20 0.34
CYP2D6 P10635 1/20 0.34
HIF1A Q16665 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
NR3C1 P04150 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5223624 0.83 SMO (0.41) PIK3CDGPR55LMNACYP1A2CYP2C19
SCHEMBL5224153 0.81 BRD4 (0.44) PIK3CDGPR55LMNACYP1A2CYP2C19
SCHEMBL5228017 0.80 SMO (0.39) PIK3CDGPR55LMNACYP1A2ALDH1A1
SCHEMBL5225729 0.78 F10 (0.38) PIK3CD
SCHEMBL5224670 0.77 NR3C1 (0.35) LMNACYP1A2ALDH1A1PTGS2NR3C1
SCHEMBL5222796 0.76 NR3C1 (0.35) LMNACYP1A2ALDH1A1PTGS2CYP3A4
SCHEMBL16404607 0.68 BRD4 (0.66) PIK3CDGPR55LMNACYP1A2CYP2C19
SCHEMBL5227271 0.67 DHODH (0.39) LMNAUSP2ALDH1A1MEN1ALOX15
SCHEMBL5227418 0.67 PTGS1 (0.38) LMNACYP2C19ALDH1A1HSD17B10CYP3A4
SCHEMBL2001301 0.67 P2RX7 (0.42) LMNACYP1A2CYP2C19ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed