SCHEMBL5223691

SCHEMBL5223691

C=CCc1cc(-c2ccc(OC)cc2)c(-c2ccc(OC)cc2)nn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
ALOX12 P18054 2/20 0.46
TP53 P04637 2/20 0.46
CYP3A4 P08684 1/20 0.46
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
CCNB2 O95067 1/20 0.40
CDK1 P06493 1/20 0.40
CCNB1 P14635 1/20 0.40
GSK3A P49840 1/20 0.40
GSK3B P49841 1/20 0.40
CDK5 Q00535 1/20 0.40
CDK5R1 Q15078 1/20 0.40
CCNB3 Q8WWL7 1/20 0.40
KMT2A Q03164 3/20 0.39
MEN1 O00255 1/20 0.39
PTGS2 P35354 2/20 0.39
MAPT P10636 2/20 0.38
NPC1 O15118 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5227512 0.77 KMT2A (0.48) SMN1; SMN2TP53KMT2AMEN1PTGS2
SCHEMBL5223978 0.74 GAA (0.50) ALDH1A1SMN1; SMN2ALOX12ALOX15KMT2A
SCHEMBL5225056 0.73 MAPK11 (0.57) ALDH1A1SMN1; SMN2KMT2AMEN1PTGS2
SCHEMBL5222119 0.72 KMT2A (0.44) ALDH1A1SMN1; SMN2TP53KMT2AMEN1
SCHEMBL5225376 0.71 ALOX5 (0.51) ALDH1A1SMN1; SMN2TP53KMT2AMEN1
SCHEMBL5677687 0.71 TP53 (0.53) ALDH1A1SMN1; SMN2ALOX12TP53CYP3A4
SCHEMBL5226722 0.71 KMT2A (0.43) ALDH1A1SMN1; SMN2TP53KMT2AMEN1
SCHEMBL5227509 0.70 MAPT (0.55) ALDH1A1SMN1; SMN2TP53TSHRKMT2A
SCHEMBL5224164 0.70 ADORA1 (0.49) ALDH1A1SMN1; SMN2TSHRKMT2AMEN1
SCHEMBL5227004 0.70 NPC1 (0.62) ALDH1A1SMN1; SMN2KMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1300399-B1 PHENYLPYRIDAZINE DERIVATIVES AND DRUGS CONTAINING THE SAME KOWA CO (JP) 2007-08-22 EP disclosed
US-6664256-B1 Interleukin- 1 beta inhibitors KOWA CO., LTD. (JP) 2003-12-16 US disclosed
EP-1300399-A1 PHENYLPYRIDAZINE DERIVATIVES AND DRUGS CONTAINING THE SAME Kowa Co., Ltd. (JP) 2003-04-09 EP disclosed