SCHEMBL5224947

SCHEMBL5224947

CCN(CC)Cc1cnn(-c2ccc(-c3ccc4c(c3)OCCO4)cc2)c1-c1ccco1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.38
HPGD P15428 5/20 0.38
PKM P14618 2/20 0.38
SIRT1 Q96EB6 2/20 0.38
CLK4 Q9HAZ1 5/20 0.38
TSHR P16473 7/20 0.38
HSD17B10 Q99714 6/20 0.38
KDM4E B2RXH2 4/20 0.38
TP53 P04637 3/20 0.38
RAB9A P51151 2/20 0.38
NPSR1 Q6W5P4 2/20 0.38
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
GAA P10253 1/20 0.38
ALOX15 P16050 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
LMNA P02545 3/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
CYP1A2 P05177 4/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224853 0.95 HSD17B10 (0.43) ALDH1A1HPGDPKMSIRT1CLK4
SCHEMBL5227284 0.90 CLK4 (0.41) ALDH1A1HPGDPKMSIRT1CLK4
SCHEMBL5229296 0.85 HSD17B10 (0.44) ALDH1A1HPGDPKMSIRT1CLK4
SCHEMBL5229195 0.85 POLB (0.40) ALDH1A1HPGDPKMSIRT1CLK4
SCHEMBL5228824 0.83 ICMT (0.40) ALDH1A1HPGDTSHRHSD17B10KDM4E
SCHEMBL5230509 0.81 POLB (0.41) ALDH1A1HPGDPKMSIRT1TSHR
SCHEMBL5224717 0.81 NPBWR1 (0.45) ALDH1A1HPGDSIRT1TSHRHSD17B10
SCHEMBL5226166 0.80 ALDH1A1 (0.41) ALDH1A1HPGDPKMSIRT1CLK4
SCHEMBL5227547 0.80 PDCD1 (0.43) ALDH1A1HPGDPKMSIRT1TSHR
SCHEMBL5228473 0.79 ALDH1A1 (0.41) ALDH1A1HPGDPKMSIRT1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed