SCHEMBL5228824

SCHEMBL5228824

CCN(CC)Cc1cnn(-c2ccc(-c3cccc(F)c3)cc2)c1-c1ccco1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ICMT O60725 1/20 0.40
NR3C1 P04150 5/20 0.38
DHODH Q02127 1/20 0.37
TP53 P04637 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TSHR P16473 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 1/20 0.35
PTGS1 P23219 1/20 0.34
PIK3R1 P27986 1/20 0.34
PIK3CA P42336 1/20 0.34
ATM Q13315 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2A Q12879 1/20 0.34
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5227271 0.90 DHODH (0.39) NR3C1DHODHTP53SMN1; SMN2TSHR
SCHEMBL5226613 0.84 SMO (0.40) NR3C1DHODHTP53SMN1; SMN2ALDH1A1
SCHEMBL5224853 0.83 HSD17B10 (0.43) TP53SMN1; SMN2TSHRALDH1A1HPGD
SCHEMBL5224717 0.83 NPBWR1 (0.45) TP53SMN1; SMN2TSHRALDH1A1HPGD
SCHEMBL5224947 0.83 ALDH1A1 (0.38) TP53SMN1; SMN2TSHRALDH1A1HPGD
SCHEMBL5229165 0.81 FLT3 (0.37) TP53SMN1; SMN2TSHRALDH1A1HPGD
SCHEMBL5230496 0.81 PTGS1 (0.37) NR3C1TP53SMN1; SMN2TSHRALDH1A1
SCHEMBL5224673 0.80 SMO (0.40) NR3C1DHODHALDH1A1PIK3R1PIK3CA
SCHEMBL2902669 0.78 ALDH1A1 (0.46) ICMTALDH1A1MEN1KMT2APIK3R1
SCHEMBL5224744 0.78 HTR1A (0.38) NR3C1DHODHTSHRALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed