SCHEMBL5223899

SCHEMBL5223899

Cn1c(-c2ccccc2N(C(=O)O)C(C)(C)C)nc2cc([N+](=O)[O-])ccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.45
PKM P14618 4/20 0.45
RAB9A P51151 2/20 0.45
RXFP1 Q9HBX9 1/20 0.45
KMT2A Q03164 6/20 0.44
LMNA P02545 5/20 0.44
KDM4E B2RXH2 1/20 0.44
MAPT P10636 1/20 0.44
APOBEC3A P31941 1/20 0.44
HTT P42858 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
APOBEC3G Q9HC16 1/20 0.44
MEN1 O00255 3/20 0.43
NPC1 O15118 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
CYP19A1 P11511 2/20 0.40
CYP2D6 P10635 1/20 0.39
PIK3CD O00329 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5225953 0.78 RAB9A (0.50) ALDH1A1PKMRAB9ARXFP1KMT2A
SCHEMBL10986929 0.75 ALDH1A1 (0.71) ALDH1A1PKMRAB9ARXFP1KMT2A
SCHEMBL3194891 0.74 ALDH1A1 (0.52) ALDH1A1PKMRAB9ARXFP1KMT2A
SCHEMBL5223908 0.74 ALDH1A1 (0.44) ALDH1A1PKMRAB9AKMT2ALMNA
SCHEMBL5225347 0.74 KDR (0.37) ALDH1A1RAB9AKDM4EMAPTNPC1
SCHEMBL5225564 0.74 KDR (0.38) ALDH1A1KDM4ECYP2D6
SCHEMBL20982763 0.71 ALDH1A1 (0.72) ALDH1A1PKMRAB9ARXFP1KMT2A
SCHEMBL5225949 0.71 ALDH1A1 (0.49) ALDH1A1PKMRAB9ARXFP1KMT2A
SCHEMBL5225943 0.71 ALDH1A1 (0.49) ALDH1A1PKMRAB9ARXFP1KMT2A
SCHEMBL1028889 0.70 L3MBTL1 (0.49) ALDH1A1LMNAMAPTHTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487824-B1 DIAMINO-PYRIMIDINES AND THEIR USE AS ANGIOGENESIS INHIBITORS SMITHKLINE BEECHAM CORP (US) 2007-06-20 EP disclosed