SCHEMBL5225922

SCHEMBL5225922

COc1ccc(-c2c(CN3CCN(C)CC3)cnn2-c2ccc(-c3ccc(F)cc3)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.53
MAPT P10636 2/20 0.53
LMNA P02545 1/20 0.53
SMO Q99835 4/20 0.53
CHKA P35790 1/20 0.47
KMT2A Q03164 1/20 0.43
PIK3CG P48736 1/20 0.43
HTR6 P50406 4/20 0.43
CYP3A4 P08684 3/20 0.43
CYP2D6 P10635 2/20 0.43
NR3C1 P04150 1/20 0.41
ALDH1A1 P00352 2/20 0.41
NPBWR1 P48145 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MAP3K11 Q16584 1/20 0.41
USP2 O75604 1/20 0.41
CYP1A2 P05177 1/20 0.41
GLA P06280 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226797 0.89 SMO (0.61) L3MBTL1MAPTLMNASMOKMT2A
SCHEMBL5224244 0.89 SMO (0.49) L3MBTL1MAPTLMNASMOCHKA
SCHEMBL5228124 0.87 SMO (0.43) L3MBTL1MAPTLMNASMO
SCHEMBL2761123 0.87 SMO (0.50) L3MBTL1MAPTLMNASMOCHKA
SCHEMBL5226795 0.83 SMO (0.42) L3MBTL1MAPTLMNASMOCHKA
SCHEMBL5227160 0.82 SMO (0.41) L3MBTL1MAPTLMNASMOCHKA
SCHEMBL5228219 0.82 SMO (0.47) L3MBTL1MAPTLMNASMOHTR6
SCHEMBL5232263 0.82 SMO (0.49) L3MBTL1MAPTLMNASMOCHKA
SCHEMBL5225265 0.81 SMO (0.59) L3MBTL1MAPTLMNASMOKMT2A
SCHEMBL5737789 0.81 SMO (0.44) L3MBTL1MAPTLMNASMOHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed