SCHEMBL5226201

SCHEMBL5226201

CC(C)CCCC(C)NC[C@@H](O)[C@H](Cc1ccsc1)N(C(=O)O)C(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.38
BACE1 P56817 1/20 0.38
BACE2 Q9Y5Z0 1/20 0.38
MME P08473 2/20 0.37
OPRM1 P35372 16/20 0.37
OPRK1 P41145 13/20 0.37
OPRD1 P41143 13/20 0.37
OPRL1 P41146 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226207 1.00 CTSD (0.38) CTSDBACE1BACE2MMEOPRM1
SCHEMBL5223660 0.82 RAB9A (0.38) CTSDBACE1BACE2CTSSCTSK
SCHEMBL5223654 0.82 RAB9A (0.38) CTSDBACE1BACE2CTSSCTSK
SCHEMBL5224498 0.80 CTSD (0.34) CTSDBACE1BACE2
SCHEMBL5224505 0.80 CTSD (0.34) CTSDBACE1BACE2
SCHEMBL5223196 0.78 CTSD (0.38) CTSDBACE1BACE2CTSSCTSK
SCHEMBL5223208 0.78 CTSD (0.38) CTSDBACE1BACE2CTSSCTSK
Hydrochloric Acid SCHEMBL5221707 0.76 CSNK1E (0.35) CTSDBACE1BACE2MMEOPRM1
SCHEMBL5221569 0.75 NPC1 (0.42) MME
SCHEMBL5221576 0.75 NPC1 (0.42) MME

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed