SCHEMBL5226314

SCHEMBL5226314

COc1ccccc1-c1c(CN2CCN(C)CC2)cnn1-c1ccc(-c2ccccc2F)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 6/20 0.46
DRD4 P21917 5/20 0.44
DRD3 P35462 4/20 0.44
DRD2 P14416 3/20 0.44
HRH2 P25021 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44
ACHE P22303 1/20 0.43
SMO Q99835 4/20 0.43
ADRA1A P35348 1/20 0.43
ALDH1A1 P00352 2/20 0.42
KDM4E B2RXH2 1/20 0.42
KMT2A Q03164 1/20 0.42
MAP4K1 Q92918 2/20 0.41
MAPK1 P28482 1/20 0.40
TGFBR1 P36897 1/20 0.39
ACVR1 Q04771 1/20 0.39
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224366 0.93 SMO (0.44) HTR7DRD4DRD3DRD2HRH2
SCHEMBL7256544 0.91 DRD4 (0.44) HTR7DRD4DRD3DRD2ACHE
SCHEMBL5226508 0.88 HTR7 (0.46) HTR7DRD4DRD3DRD2HRH2
SCHEMBL2761055 0.88 ALDH1A1 (0.46) HTR7DRD4DRD3DRD2HRH2
SCHEMBL5737789 0.87 SMO (0.44) HTR7DRD4DRD3DRD2SMO
SCHEMBL1689504 0.86 SMO (0.45) HTR7DRD4DRD3DRD2ACHE
SCHEMBL5731887 0.86 JAK2 (0.45) HTR7DRD4DRD3DRD2HRH2
SCHEMBL7261026 0.85 SMO (0.41) DRD4DRD3DRD2ACHESMO
SCHEMBL5224925 0.84 EPHB4 (0.46) HTR7DRD4DRD3DRD2ACHE
SCHEMBL5228638 0.83 DRD4 (0.41) DRD4DRD3DRD2ACHESMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed