SCHEMBL5224925

SCHEMBL5224925

COc1ccc(-c2ccc(-n3ncc(CN4CCN(C)CC4)c3-c3ccccc3F)cc2)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHB4 P54760 1/20 0.46
MCHR1 Q99705 1/20 0.40
SMO Q99835 4/20 0.40
ACHE P22303 1/20 0.38
KCNH2 Q12809 2/20 0.38
HTR7 P34969 1/20 0.38
KDM1A O60341 1/20 0.38
MAOA P21397 1/20 0.38
INSR P06213 1/20 0.37
ALK Q9UM73 1/20 0.37
DRD4 P21917 3/20 0.37
DRD3 P35462 2/20 0.37
BMPR1B O00238 2/20 0.37
ACVRL1 P37023 2/20 0.37
ACVR1 Q04771 2/20 0.37
ACVR1B P36896 1/20 0.37
RIOK2 Q9BVS4 1/20 0.37
CPB2 Q96IY4 1/20 0.36
NTRK1 P04629 1/20 0.36
CSF1R P07333 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1689504 0.88 SMO (0.45) SMOACHEHTR7DRD4DRD3
SCHEMBL5737789 0.86 SMO (0.44) SMOHTR7DRD4DRD3DRD2
SCHEMBL7256544 0.86 DRD4 (0.44) SMOACHEHTR7KDM1AMAOA
SCHEMBL2761055 0.85 ALDH1A1 (0.46) SMOACHEHTR7DRD4DRD3
SCHEMBL5226508 0.85 HTR7 (0.46) SMOACHEHTR7DRD4DRD3
SCHEMBL5228638 0.85 DRD4 (0.41) SMOACHEDRD4DRD3DRD2
SCHEMBL5226314 0.84 HTR7 (0.46) SMOACHEHTR7DRD4DRD3
SCHEMBL2761085 0.84 DHODH (0.43) SMODRD4DRD3DRD2
SCHEMBL5224217 0.84 SMO (0.44) SMOACHEALKDRD4DRD3
SCHEMBL7261049 0.84 CHKA (0.50) SMOACHEDRD4DRD3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed