SCHEMBL5226521

SCHEMBL5226521

CN(CCC#N)Cc1cnn(-c2ccc(-c3ccc(F)cc3)cc2)c1-c1ccco1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
TP53 P04637 1/20 0.35
CNKSR1 Q969H4 1/20 0.34
ALDH1A1 P00352 6/20 0.34
PGR P06401 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA2B P29275 1/20 0.34
ADORA1 P30542 1/20 0.34
NPC1 O15118 1/20 0.34
LMNA P02545 1/20 0.34
RAB9A P51151 1/20 0.34
KDM4E B2RXH2 6/20 0.33
HSD17B10 Q99714 4/20 0.33
MAPT P10636 3/20 0.33
HPGD P15428 3/20 0.33
TSHR P16473 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
GAA P10253 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5227418 0.88 PTGS1 (0.38) PTGS1SMN1; SMN2TP53ALDH1A1NPC1
SCHEMBL5226500 0.87 PTGS1 (0.36) PTGS1SMN1; SMN2TP53ALDH1A1PGR
SCHEMBL5230496 0.80 PTGS1 (0.37) PTGS1SMN1; SMN2TP53ALDH1A1NPC1
SCHEMBL13019206 0.77 PTGS1 (0.43) PTGS1SMN1; SMN2TP53CNKSR1ALDH1A1
SCHEMBL5227271 0.77 DHODH (0.39) PTGS1SMN1; SMN2TP53ALDH1A1PGR
SCHEMBL1998044 0.76 FLT3 (0.38) PTGS1SMN1; SMN2TP53ADORA2AHSD17B10
SCHEMBL1998756 0.76 NR3C1 (0.36) PTGS1SMN1; SMN2TP53ALDH1A1PGR
SCHEMBL2007394 0.75 PTGS1 (0.34) PTGS1SMN1; SMN2TP53ADORA2AMAPT
SCHEMBL5226546 0.75 ALDH1A1 (0.38) PTGS1SMN1; SMN2TP53CNKSR1ALDH1A1
SCHEMBL5224732 0.75 MAP4K4 (0.34) PTGS1SMN1; SMN2TP53ALDH1A1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed