SCHEMBL5227271

SCHEMBL5227271

CN(C)Cc1cnn(-c2ccc(-c3cccc(F)c3)cc2)c1-c1ccco1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.39
NR3C1 P04150 5/20 0.37
TP53 P04637 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TSHR P16473 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
PTGS1 P23219 1/20 0.35
PIK3R1 P27986 1/20 0.35
PIK3CA P42336 1/20 0.35
ATM Q13315 2/20 0.35
PGR P06401 2/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
ALOX15 P16050 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5228824 0.90 ICMT (0.40) DHODHNR3C1TP53SMN1; SMN2TSHR
SCHEMBL5226613 0.84 SMO (0.40) DHODHNR3C1TP53SMN1; SMN2ALDH1A1
SCHEMBL5229296 0.83 HSD17B10 (0.44) TP53SMN1; SMN2TSHRALDH1A1HPGD
SCHEMBL5226619 0.82 NPBWR1 (0.47) TP53SMN1; SMN2TSHRALDH1A1HPGD
SCHEMBL5227284 0.82 CLK4 (0.41) TP53SMN1; SMN2TSHRALDH1A1HPGD
SCHEMBL5224673 0.82 SMO (0.40) DHODHNR3C1ALDH1A1PIK3R1PIK3CA
SCHEMBL5227418 0.82 PTGS1 (0.38) NR3C1TP53SMN1; SMN2ALDH1A1HPGD
SCHEMBL5226500 0.80 PTGS1 (0.36) NR3C1TP53SMN1; SMN2ALDH1A1HPGD
SCHEMBL5224744 0.80 HTR1A (0.38) DHODHNR3C1TSHRALDH1A1HPGD
SCHEMBL5229287 0.78 EGFR (0.40) DHODHALDH1A1MEN1KMT2APTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed