SCHEMBL5226546

SCHEMBL5226546

CCC(O)c1ccccc1N(C)Cc1cnn(-c2ccc(-c3ccc(F)cc3)cc2)c1-c1ccco1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
LMNA P02545 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
PTGS1 P23219 1/20 0.33
MAPT P10636 4/20 0.33
NR3C1 P04150 3/20 0.33
TP53 P04637 2/20 0.33
NPSR1 Q6W5P4 2/20 0.32
SMO Q99835 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
FLT3 P36888 1/20 0.32
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
CASP1 P29466 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226549 0.78 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2LMNANPC1RAB9A
SCHEMBL5227418 0.78 PTGS1 (0.38) ALDH1A1SMN1; SMN2LMNANPC1RAB9A
SCHEMBL5230496 0.77 PTGS1 (0.37) ALDH1A1SMN1; SMN2LMNANPC1RAB9A
SCHEMBL13019206 0.77 PTGS1 (0.43) ALDH1A1SMN1; SMN2LMNANPC1PTGS1
SCHEMBL5226557 0.77 ALDH1A1 (0.34) ALDH1A1SMN1; SMN2LMNANPC1RAB9A
SCHEMBL5226500 0.76 PTGS1 (0.36) ALDH1A1SMN1; SMN2LMNANPC1RAB9A
SCHEMBL5226521 0.75 PTGS1 (0.35) ALDH1A1SMN1; SMN2LMNANPC1RAB9A
SCHEMBL5227271 0.74 DHODH (0.39) ALDH1A1SMN1; SMN2LMNAPTGS1NR3C1
SCHEMBL2761237 0.74 SMO (0.43) ALDH1A1SMN1; SMN2LMNAPTGS1MAPT
SCHEMBL1998044 0.73 FLT3 (0.38) SMN1; SMN2PTGS1MAPTNR3C1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed