SCHEMBL5226500

SCHEMBL5226500

CN(C)CCCN(C)Cc1cnn(-c2ccc(-c3ccc(F)cc3)cc2)c1-c1ccco1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
TP53 P04637 1/20 0.35
ALDH1A1 P00352 3/20 0.33
LMNA P02545 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
NR3C1 P04150 3/20 0.33
MAPT P10636 3/20 0.32
NPSR1 Q6W5P4 2/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
FLT3 P36888 1/20 0.32
PGR P06401 1/20 0.32
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
HPGD P15428 1/20 0.32
CASP1 P29466 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5227418 0.94 PTGS1 (0.38) PTGS1SMN1; SMN2TP53ALDH1A1LMNA
SCHEMBL5226521 0.87 PTGS1 (0.35) PTGS1SMN1; SMN2TP53ALDH1A1LMNA
SCHEMBL5230496 0.83 PTGS1 (0.37) PTGS1SMN1; SMN2TP53ALDH1A1LMNA
SCHEMBL5227271 0.80 DHODH (0.39) PTGS1SMN1; SMN2TP53ALDH1A1LMNA
SCHEMBL13019206 0.79 PTGS1 (0.43) PTGS1SMN1; SMN2TP53ALDH1A1LMNA
SCHEMBL1998044 0.78 FLT3 (0.38) PTGS1SMN1; SMN2TP53NR3C1MAPT
SCHEMBL1998756 0.77 NR3C1 (0.36) PTGS1SMN1; SMN2TP53ALDH1A1LMNA
SCHEMBL2007394 0.77 PTGS1 (0.34) PTGS1SMN1; SMN2TP53NR3C1MAPT
SCHEMBL5226619 0.76 NPBWR1 (0.47) PTGS1SMN1; SMN2TP53ALDH1A1LMNA
SCHEMBL5226546 0.76 ALDH1A1 (0.38) PTGS1SMN1; SMN2TP53ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed