SCHEMBL5226549

SCHEMBL5226549

CN(Cc1cnn(-c2ccc(-c3ccc(F)cc3)cc2)c1-c1ccco1)C(O)CCc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
RAB9A P51151 2/20 0.39
NPC1 O15118 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 2/20 0.35
TP53 P04637 2/20 0.34
SMO Q99835 1/20 0.33
NR3C1 P04150 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33
PTGS1 P23219 1/20 0.33
CNKSR1 Q969H4 1/20 0.32
UBE2I P63279 1/20 0.32
CACNA1B Q00975 1/20 0.32
APBA1 Q02410 1/20 0.32
SAE1 Q9UBE0 1/20 0.32
UBA2 Q9UBT2 1/20 0.32
TSHR P16473 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226557 0.83 ALDH1A1 (0.34) ALDH1A1SMN1; SMN2RAB9ANPC1LMNA
SCHEMBL5226546 0.78 ALDH1A1 (0.38) ALDH1A1SMN1; SMN2RAB9ANPC1LMNA
SCHEMBL5227418 0.77 PTGS1 (0.38) ALDH1A1SMN1; SMN2RAB9ANPC1LMNA
SCHEMBL13019206 0.76 PTGS1 (0.43) ALDH1A1SMN1; SMN2NPC1LMNAMAPT
SCHEMBL5226500 0.75 PTGS1 (0.36) ALDH1A1SMN1; SMN2RAB9ANPC1LMNA
SCHEMBL5230496 0.74 PTGS1 (0.37) ALDH1A1SMN1; SMN2RAB9ANPC1LMNA
SCHEMBL5226521 0.74 PTGS1 (0.35) ALDH1A1SMN1; SMN2RAB9ANPC1LMNA
SCHEMBL5227271 0.73 DHODH (0.39) ALDH1A1SMN1; SMN2LMNATP53NR3C1
SCHEMBL5224732 0.73 MAP4K4 (0.34) ALDH1A1SMN1; SMN2MAPTTP53ADORA2A
SCHEMBL5224632 0.72 ALDH1A1 (0.39) ALDH1A1SMN1; SMN2RAB9ANPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed