SCHEMBL5227096

SCHEMBL5227096

Cc1ccoc1-c1c(CN2CCN(C)CC2)cnn1-c1ccc(-c2ccc(F)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMO Q99835 4/20 0.44
DRD4 P21917 4/20 0.39
DRD3 P35462 4/20 0.39
DRD2 P14416 3/20 0.39
MAPT P10636 3/20 0.38
TNIK Q9UKE5 1/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
LMNA P02545 1/20 0.36
MAPK14 Q16539 1/20 0.35
ALDH1A1 P00352 2/20 0.35
POLB P06746 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MPO P05164 1/20 0.34
MAP4K1 Q92918 1/20 0.34
CHKA P35790 1/20 0.34
MC4R P32245 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224916 0.92 SMO (0.44) SMODRD4DRD3DRD2MAPT
SCHEMBL5228292 0.84 SMO (0.37) SMO
SCHEMBL2761009 0.83 SMO (0.43) SMODRD4DRD3DRD2MAPT
SCHEMBL1997979 0.83 SMO (0.60) SMODRD4DRD3DRD2MAPT
SCHEMBL5229176 0.82 SMO (0.39) SMODRD4DRD3DRD2MAPT
SCHEMBL5227160 0.82 SMO (0.41) SMODRD4DRD3DRD2MAPT
SCHEMBL5228124 0.80 SMO (0.43) SMODRD4DRD3DRD2MAPT
SCHEMBL5224670 0.80 NR3C1 (0.35) SMOLMNAALDH1A1NPSR1
SCHEMBL5228219 0.79 SMO (0.47) SMODRD4DRD3DRD2MAPT
SCHEMBL5224153 0.79 BRD4 (0.44) SMODRD4DRD3DRD2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed