SCHEMBL5224670

SCHEMBL5224670

Cc1ccoc1-c1c(CN(C)C)cnn1-c1ccc(-c2ccc(F)cc2)cc1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 7/20 0.35
PGR P06401 2/20 0.35
PTGS2 P35354 1/20 0.35
LMNA P02545 2/20 0.34
NPC1 O15118 1/20 0.34
ALDH1A1 P00352 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
SMO Q99835 2/20 0.33
CYP17A1 P05093 2/20 0.33
CYP1A2 P05177 2/20 0.33
NPSR1 Q6W5P4 1/20 0.32
P2RX7 Q99572 1/20 0.32
KCNH2 Q12809 1/20 0.32
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224916 0.82 SMO (0.44) LMNAALDH1A1SMONPSR1KCNH2
SCHEMBL5227096 0.80 SMO (0.44) LMNAALDH1A1SMONPSR1
SCHEMBL5222796 0.80 NR3C1 (0.35) NR3C1PGRPTGS2LMNANPC1
SCHEMBL5225124 0.77 PIK3CD (0.42) NR3C1PTGS2LMNANPC1ALDH1A1
SCHEMBL5228292 0.76 SMO (0.37) SMO
SCHEMBL5227271 0.72 DHODH (0.39) NR3C1PGRLMNAALDH1A1SMN1; SMN2
SCHEMBL5227418 0.72 PTGS1 (0.38) NR3C1LMNANPC1ALDH1A1RAB9A
SCHEMBL5229176 0.71 SMO (0.39) LMNAALDH1A1SMONPSR1
SCHEMBL5226500 0.71 PTGS1 (0.36) NR3C1PGRLMNANPC1ALDH1A1
SCHEMBL5228311 0.69 NR3C1 (0.34) NR3C1PGRLMNANPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed