SCHEMBL5229176

SCHEMBL5229176

Cc1ccoc1-c1c(CN2CCN(OC(=O)OC(C)(C)C)CC2)cnn1-c1ccc(-c2ccc(F)cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMO Q99835 4/20 0.39
THRB P10828 1/20 0.34
MAPT P10636 4/20 0.33
TP53 P04637 3/20 0.33
POLB P06746 2/20 0.33
LMNA P02545 2/20 0.33
DRD2 P14416 1/20 0.32
DRD4 P21917 1/20 0.32
DRD3 P35462 1/20 0.32
ALDH1A1 P00352 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
KDM4E B2RXH2 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
PDK2 Q15119 1/20 0.31
SSTR5 P35346 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5227096 0.82 SMO (0.44) SMOMAPTPOLBLMNADRD2
SCHEMBL5224916 0.82 SMO (0.44) SMOMAPTTP53POLBLMNA
SCHEMBL5226151 0.80 SMO (0.35) SMOTP53LMNAALDH1A1KDM4E
SCHEMBL5228292 0.76 SMO (0.37) SMO
SCHEMBL5226715 0.75 ALDH1A1 (0.37) THRBMAPTTP53POLBLMNA
SCHEMBL5224994 0.75 MAPT (0.35) THRBMAPTTP53POLBLMNA
SCHEMBL5224670 0.71 NR3C1 (0.35) SMOLMNAALDH1A1NPSR1
SCHEMBL5227160 0.67 SMO (0.41) SMOMAPTLMNADRD2DRD4
SCHEMBL5225508 0.67 SSTR5 (0.36) SMOTHRBMAPTTP53LMNA
SCHEMBL2761009 0.67 SMO (0.43) SMOMAPTTP53LMNADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed