SCHEMBL5230316

SCHEMBL5230316

O=[N+]([O-])c1csc(S(=O)(=O)Nc2ccc(Cl)cc2)c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CES1 P23141 1/20 0.49
IDH1 O75874 4/20 0.45
KDM1A O60341 2/20 0.44
CA2 P00918 3/20 0.43
CA1 P00915 2/20 0.43
CA12 O43570 1/20 0.42
CA9 Q16790 1/20 0.42
MAPT P10636 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CYP19A1 P11511 1/20 0.41
MCL1 Q07820 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5230151 0.76 CES1 (0.73) CES1KDM1ACA2CA1CA12
SCHEMBL5237280 0.75 CES1 (0.49) CES1IDH1MAPTMEN1KMT2A
SCHEMBL5229246 0.74 MEN1 (0.52) CES1IDH1CA2CA1MAPT
SCHEMBL5228114 0.73 ALDH1A1 (0.71) CES1IDH1KDM1ACA2CA1
SCHEMBL5228629 0.73 IDH1 (0.51) CES1IDH1MAPTNPSR1MEN1
SCHEMBL23832701 0.72 IDH1 (0.54) CES1IDH1CA2CA1MAPT
SCHEMBL30218156 0.72 IDH1 (0.54) CES1IDH1CA2CA1MAPT
SCHEMBL18228 0.72 ALDH1A1 (0.36) CA2CA1CA12CA9MEN1
SCHEMBL7580547 0.71 IDH1 (0.71) IDH1MCL1
SCHEMBL5228023 0.71 CA2 (0.49) CA2CA1CA12CA9MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1519932-B1 BISARYLSULFONAMIDE COMPOUNDS AND THEIR USE IN CANCER THERAPY CYCLACEL LTD (GB) 2007-10-03 EP claimed
EP-1519932-B1 BISARYLSULFONAMIDE COMPOUNDS AND THEIR USE IN CANCER THERAPY CYCLACEL LTD (GB) 2007-10-03 EP disclosed