SCHEMBL5239459

SCHEMBL5239459

CC(C)N(c1nn(-c2ccc(Cl)cc2)cc1OC(=O)O)C(=O)[C@H]1CC[C@H](C)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
KMT2A Q03164 2/20 0.33
BLM P54132 1/20 0.33
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
HRH3 Q9Y5N1 4/20 0.31
TRPV1 Q8NER1 1/20 0.31
CNR1 P21554 1/20 0.31
KCNH2 Q12809 1/20 0.31
CYP1A2 P05177 1/20 0.31
HIF1A Q16665 1/20 0.31
MET P08581 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
MAPT P10636 1/20 0.31
PKM P14618 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5231776 0.92 ESRRA (0.32) KDM4ENPC1RAB9AKMT2ACYP1A2
SCHEMBL5236797 0.91
SCHEMBL5236128 0.91 NPC1 (0.34) KDM4ENPC1RAB9AKMT2ACA12
SCHEMBL5233446 0.91 NPC1 (0.35) KDM4ENPC1RAB9AKMT2AALDH1A1
SCHEMBL5234344 0.90 ESRRA (0.31)
SCHEMBL5231417 0.90 HRH3 (0.36) KDM4EKMT2AHRH3TRPV1ALDH1A1
SCHEMBL5233835 0.89 KCNJ1 (0.32) KMT2AALDH1A1MAPT
SCHEMBL5234129 0.89 ADORA3 (0.37) KDM4EKMT2ACA12CA1CA2
SCHEMBL5232934 0.89 KDM4E (0.30) KDM4EALDH1A1
SCHEMBL5238208 0.89 ALDH1A1 (0.38) KDM4ENPC1RAB9ACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730116-B1 4-CARBOX PYRAZOLE DERIVATES USEFUL AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORP (US) 2007-09-05 EP claimed