SCHEMBL5235487

SCHEMBL5235487

O=C(Cc1ccnc2ccccc12)c1cc(F)cc(C(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.44
VNN1 O95497 4/20 0.44
AURKA O14965 1/20 0.43
TACR1 P25103 2/20 0.42
CNR2 P34972 2/20 0.40
KDR P35968 3/20 0.40
BRAF P15056 1/20 0.40
MAPK14 Q16539 1/20 0.40
TNNI3K Q59H18 1/20 0.40
FLT1 P17948 1/20 0.40
NR2E1 Q9Y466 2/20 0.39
RIPK1 Q13546 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.38
CYP3A4 P08684 1/20 0.38
GPBAR1 Q8TDU6 1/20 0.38
RORA P35398 1/20 0.38
PIK3CA P42336 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5233508 0.85 CNR2 (0.53) CYP1A2VNN1CNR2KDRBRAF
SCHEMBL5239397 0.84 CNR2 (0.50) CYP1A2TACR1CNR2KDRBRAF
SCHEMBL5235758 0.83 AURKA (0.39) CYP1A2VNN1AURKATACR1CNR2
SCHEMBL5235754 0.83 AURKA (0.39) CYP1A2VNN1AURKATACR1CNR2
SCHEMBL5231753 0.81 CYP1A2 (0.53) CYP1A2LOXL2CYP3A4
SCHEMBL5237313 0.79 RAB9A (0.56) CYP1A2LOXL2CYP3A4
SCHEMBL5239743 0.79 VNN1 (0.44) CYP1A2VNN1KDRRIPK1LOXL2
SCHEMBL5239658 0.76 CYP1A2 (0.61) CYP1A2LOXL2CYP3A4
SCHEMBL29987166 0.76 CYP1A2 (0.61) CYP1A2LOXL2CYP3A4
SCHEMBL5239559 0.73 KAT6A (0.44) CYP1A2KDRBRAFMAPK14TNNI3K

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed