SCHEMBL5239743

SCHEMBL5239743

O=C(Cc1ccnc2ccccc12)c1ccc(F)c(C(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 7/20 0.44
CYP1A2 P05177 1/20 0.44
KMO O15229 1/20 0.41
GRM4 Q14833 1/20 0.41
RIPK1 Q13546 1/20 0.40
CETP P11597 1/20 0.39
KCNQ3 O43525 1/20 0.39
KCNQ2 O43526 1/20 0.39
KCNE1 P15382 1/20 0.39
KCNQ1 P51787 1/20 0.39
KDR P35968 1/20 0.39
NR3C2 P08235 1/20 0.38
LOXL2 Q9Y4K0 1/20 0.38
AR P10275 1/20 0.38
GPBAR1 Q8TDU6 1/20 0.38
RPS6KB1 P23443 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5239397 0.81 CNR2 (0.50) CYP1A2KDRLOXL2
SCHEMBL5233508 0.81 CNR2 (0.53) VNN1CYP1A2KDR
SCHEMBL5237313 0.79 RAB9A (0.56) CYP1A2LOXL2
SCHEMBL5231753 0.79 CYP1A2 (0.53) CYP1A2GRM4LOXL2AR
SCHEMBL5235487 0.79 CYP1A2 (0.44) VNN1CYP1A2RIPK1KDRLOXL2
SCHEMBL5235891 0.77 CYP1A2 (0.45) CYP1A2KDRLOXL2GPBAR1RPS6KB1
SCHEMBL5233678 0.77 RAB9A (0.56) CYP1A2KDRLOXL2
SCHEMBL5238619 0.76 KDR (0.35) VNN1CYP1A2KDRAR
SCHEMBL5234876 0.76 CYP1A2 (0.49) CYP1A2KDRLOXL2
SCHEMBL5239658 0.76 CYP1A2 (0.61) CYP1A2LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed