SCHEMBL5239397

SCHEMBL5239397

O=C(Cc1ccnc2ccccc12)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 1/20 0.50
CYP1A2 P05177 1/20 0.49
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
PTPN1 P18031 2/20 0.45
GSK3B P49841 1/20 0.45
BCHE P06276 1/20 0.44
HSD11B1 P28845 1/20 0.44
LOXL2 Q9Y4K0 1/20 0.43
TLR7 Q9NYK1 1/20 0.43
KDM4E B2RXH2 1/20 0.42
GLA P06280 1/20 0.42
PDPK1 O15530 1/20 0.42
PTGDR2 Q9Y5Y4 1/20 0.42
TACR1 P25103 1/20 0.41
KDR P35968 2/20 0.41
BRAF P15056 1/20 0.41
MAPK14 Q16539 1/20 0.41
TNNI3K Q59H18 1/20 0.41
FLT1 P17948 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5233508 0.86 CNR2 (0.53) CNR2CYP1A2TLR7KDRBRAF
SCHEMBL5237313 0.85 RAB9A (0.56) CYP1A2MEN1KMT2APTPN1LOXL2
SCHEMBL5239658 0.84 CYP1A2 (0.61) CYP1A2MEN1KMT2APTPN1LOXL2
SCHEMBL29987166 0.84 CYP1A2 (0.61) CYP1A2MEN1KMT2APTPN1LOXL2
SCHEMBL5235487 0.84 CYP1A2 (0.44) CNR2CYP1A2LOXL2TACR1KDR
SCHEMBL5233678 0.82 RAB9A (0.56) CYP1A2MEN1KMT2ALOXL2KDM4E
SCHEMBL5239743 0.81 VNN1 (0.44) CYP1A2LOXL2KDR
SCHEMBL5237502 0.81 LOXL2 (0.43) CNR2CYP1A2BCHELOXL2PTGDR2
SCHEMBL5235015 0.81 LOXL2 (0.43) CNR2CYP1A2BCHELOXL2PTGDR2
SCHEMBL17583692 0.79 TDP1 (0.53) CNR2MEN1KMT2APTPN1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed