SCHEMBL5236137

SCHEMBL5236137

COc1ccc(-c2c(C3CCCCC3)c3sc(OC(=O)O)cc3n2CC(=O)N2CCOCC2)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 2/20 0.46
GRIN2B Q13224 2/20 0.46
PTGS2 P35354 3/20 0.45
USP2 O75604 1/20 0.42
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
TP53 P04637 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
FKBP1A P62942 2/20 0.41
CNR2 P34972 1/20 0.40
POLB P06746 2/20 0.40
GAA P10253 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5234725 0.93 EGFR (0.42) GRIN1GRIN2BPTGS2USP2RAB9A
SCHEMBL5230063 0.92 EGFR (0.41) GRIN1GRIN2BPTGS2TP53HSD17B10
SCHEMBL5238339 0.91 MAPK1 (0.42) GRIN1GRIN2BPTGS2USP2NPC1
SCHEMBL5230369 0.90 ALDH1A1 (0.38) GRIN1GRIN2BPTGS2KDM4EALDH1A1
SCHEMBL424159 0.89 GRIN1 (0.46) GRIN1GRIN2BPTGS2USP2NPC1
SCHEMBL5231149 0.89 GRIN2B (0.39) GRIN1GRIN2BPTGS2NPC1RAB9A
SCHEMBL5233368 0.88 LMNA (0.39) GRIN1GRIN2BPOLBGAAL3MBTL1
SCHEMBL5232857 0.86 FKBP1A (0.38) GRIN2BNPC1RAB9ATP53SMN1; SMN2
SCHEMBL5434937 0.80 PTGS2 (0.46) GRIN1GRIN2BPTGS2USP2NPC1
SCHEMBL2996624 0.80 MAPK1 (0.44) GRIN2BUSP2NPC1RAB9ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664059-B1 THIENOPYRROLES AS ANTIVIRAL AGENTS ANGELETTI P IST RICHERCHE BIO (IT) 2007-09-12 EP claimed