Hydroxyamine

Hydroxyamine

SCHEMBL5236480

NO.O=C(O)[C@H]1CCN1C(=S)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.43
GAA P10253 2/20 0.40
CES2 O00748 1/20 0.40
RHOC P08134 4/20 0.39
RHOA P61586 4/20 0.39
HIF1A Q16665 1/20 0.39
CYP3A4 P08684 3/20 0.38
TSHR P16473 1/20 0.38
CNR1 P21554 1/20 0.38
USP2 O75604 4/20 0.37
CYP2C9 P11712 4/20 0.37
HSD17B10 Q99714 2/20 0.37
TDP1 Q9NUW8 1/20 0.36
CYP2C19 P33261 2/20 0.36
POLB P06746 1/20 0.36
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3548143 0.83 RHOA (0.45) TACR1GAACES2RHOCRHOA
SCHEMBL3544517 0.82 PDK2 (0.44) TACR1GAACES2RHOCRHOA
SCHEMBL5271173 0.82 PDK2 (0.44) TACR1GAACES2RHOCRHOA
Hydroxyamine SCHEMBL5238906 0.80 LMNA (0.50) CES2POLB
Hydroxyamine SCHEMBL5238910 0.80 LMNA (0.50) CES2POLB
SCHEMBL5201383 0.77 LMNA (0.40) CES2POLB
Hydroxyamine SCHEMBL5270947 0.75 CACNA1B (0.36) CYP2C9HSD17B10CYP2C19
Hydroxyamine SCHEMBL5270943 0.75 CACNA1B (0.36) CYP2C9HSD17B10CYP2C19
SCHEMBL1534220 0.75 RHOC (0.62) TACR1RHOCRHOATDP1
SCHEMBL3552980 0.74 ADCY8 (0.42) GAARHOACYP3A4CNR1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539744-A4 N-HYDROXYAMIDE DERIVATIVES POSSESSING ANTIBACTERIAL ACTIVITY VICURON PHARM INC (US) 2007-06-06 EP disclosed
EP-1539744-A2 N-HYDROXYAMIDE DERIVATIVES POSSESSING ANTIBACTERIAL ACTIVITY Vicuron Pharmaceuticals, Inc. (US) 2005-06-15 EP disclosed
WO-2004007444-A2 N-HYDROXYAMIDE DERIVATIVES POSSESSING ANTIBACTERIAL ACTIVITY VICURON PHARMACEUTICALS, INC. (US) 2004-01-22 WO disclosed