SCHEMBL5236808

SCHEMBL5236808

Cc1ccc(C(Br)C=O)c2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.48
CYP2A6 P11509 3/20 0.38
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35
PABPC1 P11940 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ALDH1A1 P00352 3/20 0.33
TSHR P16473 2/20 0.32
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
GRIN2C Q14957 1/20 0.32
GRIN3A Q8TCU5 1/20 0.32
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9319118 0.78 CYP1A2 (0.59) CYP1A2CYP2A6KDM4EMAPTPABPC1
SCHEMBL5241189 0.78 ALDH1A1 (0.32) CYP1A2ALDH1A1TSHRCYP2C9CYP2C19
SCHEMBL5949775 0.77 IMPDH2 (0.45) CYP1A2KDM4EMAPTALDH1A1CYP2C9
SCHEMBL168886 0.76 ESR1 (0.45) MAPTALDH1A1TSHRGRIN2DGRIN3B
SCHEMBL7007166 0.73 CYP1A2 (0.65) CYP1A2CYP2A6KDM4EMAPTPABPC1
SCHEMBL845776 0.73 ALDH1A1 (0.61) CYP1A2CYP2A6ALDH1A1TSHRCYP2C9
SCHEMBL5949824 0.72 PARP1 (0.39) CYP1A2ALDH1A1CYP2C9CYP2C19
SCHEMBL6619213 0.71 CYP1A2 (0.46) CYP1A2CYP2A6KDM4EMAPTALDH1A1
SCHEMBL7833173 0.71 CYP1A2 (0.62) CYP1A2CYP2A6KDM4EMAPTPABPC1
SCHEMBL5236200 0.70 CYP1A2 (0.48) CYP1A2CYP2A6KDM4EALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1851232-A2 DIHYDROIMIDAZOTHIAZOLE DERIVATIVES Prosidion Limited (GB) 2007-11-07 EP disclosed
WO-2006085118-A2 DIHYDROIMIDAZOTHIAZOLE DERIVATIVES PROSIDION LIMITED (GB) 2006-08-17 WO disclosed