SCHEMBL5241189

SCHEMBL5241189

O=CC(Br)c1ccc(F)c2ccccc12

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.32
TSHR P16473 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
SIGMAR1 Q99720 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5236808 0.78 CYP1A2 (0.48) ALDH1A1TSHRCYP1A2CYP2C9CYP2C19
SCHEMBL20551403 0.76 CES2 (0.40) ALDH1A1CYP2C9
SCHEMBL166430 0.76 CES2 (0.40) ALDH1A1CYP2C9
SCHEMBL5949775 0.74 IMPDH2 (0.45) ALDH1A1CYP1A2CYP2C9
SCHEMBL845776 0.73 ALDH1A1 (0.61) ALDH1A1TSHRCYP1A2CYP2C9CYP2C19
SCHEMBL5949824 0.72 PARP1 (0.39) ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL20551784 0.71
SCHEMBL20551400 0.70 MDM2 (0.38)
SCHEMBL5236200 0.70 CYP1A2 (0.48) ALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL12463310 0.70 HTR2B (0.42) ALDH1A1TSHRCYP1A2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1851232-A2 DIHYDROIMIDAZOTHIAZOLE DERIVATIVES Prosidion Limited (GB) 2007-11-07 EP disclosed
WO-2006085118-A2 DIHYDROIMIDAZOTHIAZOLE DERIVATIVES PROSIDION LIMITED (GB) 2006-08-17 WO disclosed
EP-1648876-A1 5-HT SB 2B /SB RECEPTOR ANTAGONISTS Pharmagene Laboratories Ltd (GB) 2006-04-26 EP disclosed
WO-2005012263-A1 5-HT2B RECEPTOR ANTAGONISTS PHARMAGENE LABORATORIES LIMITED (GB) 2005-02-10 WO disclosed