SCHEMBL5236897

SCHEMBL5236897

CNC(=O)COC(=O)N1CCN(c2ccccc2Oc2ccccc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.53
TSHR P16473 5/20 0.53
GAA P10253 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
NPSR1 Q6W5P4 3/20 0.47
MAPT P10636 5/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
HTR1A P08908 1/20 0.46
SLC6A2 P23975 1/20 0.46
SLC6A4 P31645 1/20 0.46
SLC6A3 Q01959 1/20 0.46
LMNA P02545 4/20 0.45
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
PKM P14618 1/20 0.44
HSD17B10 Q99714 2/20 0.44
TP53 P04637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5239273 0.87 ALDH1A1 (0.60) ALDH1A1TSHRMEN1KMT2ALMNA
SCHEMBL5235199 0.82 GAA (0.53) ALDH1A1TSHRGAASMN1; SMN2NPSR1
SCHEMBL5232433 0.82 ALDH1A1 (0.59) ALDH1A1TSHRGAASMN1; SMN2NPSR1
SCHEMBL5233076 0.81 GAA (0.50) ALDH1A1GAASMN1; SMN2MAPTMEN1
SCHEMBL5234580 0.81 GAA (0.46) ALDH1A1TSHRGAASMN1; SMN2CYP1A2
SCHEMBL5237576 0.81 KMT2A (0.53) ALDH1A1TSHRGAASMN1; SMN2NPSR1
SCHEMBL5239407 0.80 MAPT (0.52) ALDH1A1TSHRGAASMN1; SMN2NPSR1
SCHEMBL5235922 0.79 HTR1A (0.51) ALDH1A1GAASMN1; SMN2MAPTKMT2A
SCHEMBL5237366 0.78 AKR1C3 (0.52) ALDH1A1GAASMN1; SMN2MAPT
SCHEMBL5234799 0.78 MAPT (0.74) ALDH1A1TSHRGAASMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1701946-B1 DERIVATIVES OF 1-PIPERAZINE- AND 1-HOMOPIPERAZINE-CARBOXYLATES, PREPARATION METHOD THEREOF AND USE OF SAME AS INHIBITORS OF THE FAAH ENZYME SANOFI AVENTIS (FR) 2007-12-19 EP claimed