SCHEMBL5237329

SCHEMBL5237329

CNC1(CC=O)CN(c2ccc(C(F)(F)F)cc2)CCN1C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.40
CA12 O43570 1/20 0.40
CA9 Q16790 1/20 0.40
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
AKR1C3 P42330 1/20 0.39
NOTUM Q6P988 1/20 0.39
PPARD Q03181 4/20 0.38
PPARA Q07869 3/20 0.38
DEGS1 O15121 1/20 0.38
ME2 P23368 1/20 0.38
ME1 P48163 1/20 0.38
ME3 Q16798 1/20 0.38
PTGES O14684 2/20 0.37
MAPT P10636 2/20 0.37
LMNA P02545 1/20 0.37
MMP2 P08253 1/20 0.36
MMP3 P08254 1/20 0.36
MMP9 P14780 1/20 0.36
MMP8 P22894 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5233790 0.97 CA2 (0.38) CA2CA12CA9DRD2DRD4
SCHEMBL5232294 0.88 ALDH1A1 (0.39) CA2CA12CA9MAPTLMNA
SCHEMBL5232337 0.88 LMNA (0.45) NOTUMMAPTLMNASMN1; SMN2
SCHEMBL5232205 0.88 SLC6A7 (0.41) MAPTLMNASMN1; SMN2
SCHEMBL5239788 0.86 MAPT (0.43) AKR1C3MAPTLMNASMN1; SMN2
SCHEMBL5238192 0.86 CYP2C19 (0.37) MAPTLMNA
SCHEMBL5230481 0.85 ITGB3 (0.39)
SCHEMBL5234847 0.85 KMT2A (0.40) CA2CA12CA9MAPTLMNA
SCHEMBL5236555 0.84 USP2 (0.41) MAPTTP53SMN1; SMN2
SCHEMBL5237663 0.84 KCNA5 (0.37) PPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1701946-B1 DERIVATIVES OF 1-PIPERAZINE- AND 1-HOMOPIPERAZINE-CARBOXYLATES, PREPARATION METHOD THEREOF AND USE OF SAME AS INHIBITORS OF THE FAAH ENZYME SANOFI AVENTIS (FR) 2007-12-19 EP claimed