SCHEMBL5237685

SCHEMBL5237685

Cc1cccc(C(=O)Cc2cccnc2)n1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.53
IDO1 P14902 13/20 0.51
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C9 P11712 1/20 0.48
P2RX7 Q99572 1/20 0.46
CYP2A6 P11509 1/20 0.46
GRM5 P41594 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2801582 0.83 P2RX7 (0.53) P2RX7GRM5
SCHEMBL5240146 0.78 RAB9A (0.57) P2RX7GRM5
SCHEMBL18230341 0.77 HTT (0.62) NAPRTIDO1CYP1A2CYP3A4CYP2C9
SCHEMBL5198154 0.77 P2RX7 (0.46) CYP1A2P2RX7GRM5
SCHEMBL5235569 0.76 P2RX7 (0.49) P2RX7GRM5
SCHEMBL4030946 0.74 HDAC3 (0.49) P2RX7
SCHEMBL6283045 0.74 IDO1 (0.58) NAPRTIDO1CYP1A2CYP3A4CYP2C9
SCHEMBL5240771 0.73 USP2 (0.51) CYP3A4P2RX7
SCHEMBL5235128 0.73 ALOX5 (0.49) CYP1A2P2RX7CYP2A6GRM5
SCHEMBL3281175 0.73 VNN1 (0.58) NAPRTIDO1CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed