SCHEMBL5243554

SCHEMBL5243554

COc1ccc(CN(CC(=O)O)c2ccccc2Cl)c(OC)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.48
KDM4E B2RXH2 5/20 0.48
TSHR P16473 2/20 0.48
POLB P06746 2/20 0.47
HTT P42858 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
LMNA P02545 2/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
KMT2A Q03164 3/20 0.47
MEN1 O00255 2/20 0.47
TDP1 Q9NUW8 2/20 0.46
BCL2A1 Q16548 1/20 0.43
HSD17B10 Q99714 1/20 0.42
TSPO P30536 1/20 0.42
HTR2A P28223 1/20 0.42
SLC6A4 P31645 1/20 0.42
KCNH2 Q12809 1/20 0.42
TAS1R3 Q7RTX0 1/20 0.42
TAS1R1 Q7RTX1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21246777 0.79 TSPO (0.49) ALDH1A1KDM4ETSHRPOLBKMT2A
SCHEMBL4841869 0.77 MEN1 (0.52) ALDH1A1KDM4ETSHRPOLBHTT
SCHEMBL5209687 0.74 ALDH1A1 (0.46) ALDH1A1KDM4ETSHRPOLBHTT
SCHEMBL30465852 0.74 APLNR (0.51) ALDH1A1KDM4ETSHRPOLBHTT
SCHEMBL341820 0.73 TDP1 (0.56) ALDH1A1SMN1; SMN2KMT2AMEN1TDP1
SCHEMBL7576003 0.70 TSPO (0.71) TSPO
SCHEMBL6582986 0.70 TDP1 (0.48) ALDH1A1KDM4ETSHRPOLBHTT
SCHEMBL1097902 0.69 HSD17B10 (0.75) ALDH1A1KDM4EPOLBKMT2AMEN1
SCHEMBL30831943 0.69 HSD17B10 (0.75) ALDH1A1KDM4EPOLBKMT2AMEN1
SCHEMBL3651761 0.69 TDP1 (0.70) TSHRPOLBHTTSMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343561-B1 SERINE PROTEASE INHIBITORS TULARIK LTD (GB) 2007-02-28 EP disclosed