SCHEMBL5244571

SCHEMBL5244571

Cc1ccsc1CNC(=O)c1nnn(-c2ccc(C(=O)NCC(F)(F)F)cc2)c1COCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.41
CCR1 P32246 1/20 0.40
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
HPGD P15428 2/20 0.37
POLB P06746 1/20 0.36
LMNA P02545 2/20 0.36
EPHX2 P34913 1/20 0.35
MIF P14174 2/20 0.35
TP53 P04637 1/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
GABRA5 P31644 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PTGER1 P34995 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5250048 0.88 EPHX2 (0.46) CCR1MEN1KMT2AHPGDLMNA
SCHEMBL5245240 0.87 HPGD (0.45) MAOACCR1MEN1KMT2AHPGD
SCHEMBL5244539 0.86 SMO (0.44) CCR1MEN1KMT2AHPGDLMNA
SCHEMBL5248134 0.85 P2RX3 (0.42) CCR1MEN1KMT2AHPGDLMNA
SCHEMBL5248045 0.85 GRM5 (0.43) CCR1MEN1KMT2AHPGDLMNA
SCHEMBL5247431 0.85 RIPK1 (0.44) CCR1MEN1KMT2AHPGDLMNA
SCHEMBL5245587 0.84 RAB9A (0.49) MAOACCR1MEN1KMT2ALMNA
SCHEMBL5245586 0.84 CCR1 (0.46) CCR1MEN1KMT2AHPGDLMNA
SCHEMBL5244893 0.84 MAPK14 (0.48) MAOACCR1EPHX2HDAC1
Trifluoroacetic Acid SCHEMBL5246743 0.83 MAPK14 (0.44) MEN1KMT2AHPGDPOLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed