SCHEMBL5246379

SCHEMBL5246379

CCNC(=O)c1ccc(-n2nnc(C(=O)NCc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c2CSC)cc1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 2/20 0.50
CCR1 P32246 2/20 0.49
HPGD P15428 6/20 0.45
ALDH1A1 P00352 6/20 0.45
KDM4E B2RXH2 4/20 0.45
CYP1A2 P05177 3/20 0.45
CYP2D6 P10635 3/20 0.45
CYP2C19 P33261 3/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
LMNA P02545 2/20 0.44
GAA P10253 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
RECQL P46063 1/20 0.41
HDAC1 Q13547 1/20 0.39
P2RY14 Q15391 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5247130 0.95 CCR1 (0.46) MLYCDCCR1HPGDALDH1A1KDM4E
SCHEMBL5246999 0.93 HDAC1 (0.46) CCR1ALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL5244318 0.92 CCR1 (0.59) MLYCDCCR1CYP1A2CYP2D6CYP2C19
SCHEMBL5249308 0.88 RIPK1 (0.46) CCR1HPGDALDH1A1CYP1A2CYP2C19
SCHEMBL5246092 0.86 EPHX2 (0.53) CYP1A2CYP2C19LMNA
SCHEMBL5248524 0.86 LMNA (0.43) MLYCDCCR1CYP1A2CYP2D6CYP2C19
SCHEMBL5244456 0.85 LMNA (0.57) ALDH1A1LMNAHDAC1
SCHEMBL5244694 0.85 HPGD (0.48) HPGDALDH1A1KDM4ECYP1A2CYP2C19
Trifluoroacetic Acid SCHEMBL5247370 0.85 LMNA (0.48) HPGDALDH1A1CYP1A2CYP2D6CYP2C19
SCHEMBL5245295 0.85 LMNA (0.44) CCR1HPGDALDH1A1CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed
EP-1763303-A1 SUBSTITUTED PYRIDAZINE CARBOXAMIDES AND DERIVATIVES THEREOF Bayer CropScience Aktiengesellschaft (DE) 2007-03-21 EP disclosed
WO-2006000333-A1 SUBSTITUTED PYRIDAZINE CARBOXAMIDES AND DERIVATIVES THEREOF BAYER CROPSCIENCE AKTIENGESELLSCHAFT (DE) 2006-01-05 WO disclosed