SCHEMBL5249308

SCHEMBL5249308

CCNC(=O)c1ccc(-n2nnc(C(=O)NCc3cc(F)cc(F)c3)c2CSC)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.46
LMNA P02545 2/20 0.46
EGLN1 Q9GZT9 1/20 0.41
MAPT P10636 3/20 0.39
CCR1 P32246 1/20 0.39
HPGD P15428 2/20 0.38
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
RECQL P46063 1/20 0.38
SMO Q99835 1/20 0.38
AURKA O14965 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ROCK2 O75116 1/20 0.36
ROCK1 Q13464 1/20 0.36
BRD4 O60885 1/20 0.36
MIF P14174 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5247130 0.92 CCR1 (0.46) RIPK1LMNACCR1HPGDALDH1A1
SCHEMBL5244366 0.92 CCR1 (0.45) RIPK1LMNAMAPTCCR1ALDH1A1
SCHEMBL5244456 0.91 LMNA (0.57) LMNAMAPTALDH1A1SMOMIF
SCHEMBL5245295 0.89 LMNA (0.44) LMNAMAPTCCR1HPGDALDH1A1
SCHEMBL5246379 0.88 MLYCD (0.50) LMNACCR1HPGDALDH1A1CYP1A2
SCHEMBL5244694 0.87 HPGD (0.48) LMNAMAPTHPGDALDH1A1CYP1A2
SCHEMBL5244114 0.87 CCR1 (0.43) LMNAMAPTCCR1HPGDALDH1A1
SCHEMBL5245644 0.86 LMNA (0.41) LMNAMAPTCCR1HPGDALDH1A1
SCHEMBL5247031 0.86 LMNA (0.41) LMNAHPGDALDH1A1CYP1A2CYP2C9
SCHEMBL5249263 0.86 LMNA (0.45) LMNACCR1HPGDALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed