SCHEMBL525342

SCHEMBL525342

Oc1nc2ccccc2c(I)c1Cl

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.52
MAOB P27338 1/20 0.52
KDM4E B2RXH2 6/20 0.38
ALDH1A1 P00352 5/20 0.38
GLA P06280 4/20 0.38
HPGD P15428 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
TDP1 Q9NUW8 3/20 0.38
GAA P10253 3/20 0.38
CASP1 P29466 2/20 0.38
CASP7 P55210 2/20 0.38
HSD17B10 Q99714 2/20 0.38
ATM Q13315 2/20 0.38
CHRM2 P08172 1/20 0.38
ADRA2A P08913 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
CHRM1 P11229 1/20 0.38
NQO2 P16083 1/20 0.38
DRD1 P21728 1/20 0.38
ACHE P22303 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10527280 0.85 MAOA (0.57) MAOAMAOBKDM4EALDH1A1GLA
SCHEMBL44256 0.82 KDM4E (0.41) MAOAMAOBKDM4EALDH1A1GLA
SCHEMBL28961139 0.82 MAOA (0.64) MAOAMAOBKDM4EALDH1A1GLA
SCHEMBL31413138 0.77 MAOA (0.52) MAOAMAOBKDM4EALDH1A1GLA
SCHEMBL13445183 0.74 KDM4E (0.56) MAOAMAOBKDM4EALDH1A1GLA
SCHEMBL10527277 0.73 MAOA (0.47) MAOAMAOBKDM4EALDH1A1GLA
SCHEMBL667261 0.73 MAOA (0.52) MAOAMAOBKDM4EALDH1A1GLA
SCHEMBL7552792 0.73 GPR3 (0.44) MAOAKDM4EALDH1A1GLAHPGD
SCHEMBL5349939 0.72 MAOA (0.61) MAOAMAOBKDM4EALDH1A1GLA
SCHEMBL7607540 0.70 GPR3 (0.54) MAOAMAOBKDM4EALDH1A1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 179 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4539816-A1 COMPOSITIONS AND METHODS FOR AN ORAL SUPPLEMENT TO ORAL MINOXIDIL FOR THE TREATMENT OF ALOPECIA Follea International (US) 2025-04-23 EP claimed
WO-2025048828-A1 COMPOSITIONS AND METHODS FOR AN ORAL SUPPLEMENT TO ORAL MINOXIDIL FOR THE TREATMENT OF ALOPECIA FOLLEA INTERNATIONAL (US) 2025-03-06 WO claimed
EP-3720468-B1 TISSUE REPAIR UNIV SUSSEX (GB) 2024-10-30 EP claimed
US-11596668-B2 Tissue repair THE UNIVERSITY OF SUSSEX (GB) 2023-03-07 US claimed
US-20210162008-A1 TISSUE REPAIR THE UNIVERSITY OF SUSSEX (GB) 2021-06-03 US claimed
EP-3720468-A1 TISSUE REPAIR The University of Sussex (GB) 2020-10-14 EP claimed
WO-2019110999-A1 TISSUE REPAIR THE UNIVERSITY OF SUSSEX (GB) 2019-06-13 WO claimed
US-20160206579-A1 TAURINE OR TAURINE-LIKE SUBSTANCES FOR THE PREVENTION AND TREATMENT OF A DISEASE ASSOCIATED WITH RETINAL GANGLION CELL DEGENERATION INSERM (Institut National de la Santé et de la Recherche Médicale) (FR) 2016-07-21 US claimed
US-20120027723-A1 TAURINE OR TAURINE-LIKE SUBSTANCES FOR THE PREVENTION AND TREATMENT OF A DISEASE ASSOCIATED WITH RETINAL GANGLION CELL DEGENERATION INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 2012-02-02 US claimed
EP-2393490-A1 TAURINE OR TAURINE-LIKE SUBSTANCES FOR THE PREVENTION AND TREATMENT OF A DISEASE ASSOCIATED WITH RETINAL GANGLION CELL DEGENERATION INSERM - Institut National de la Santé et de la Recherche Médicale (FR) 2011-12-14 EP claimed
CN-102274347-A Anticancer composition and application thereof 2011-12-14 CN claimed
WO-2011113904-A1 MEDICAMENTS FOR THE PREVENTION AND TREATMENT OF A DISEASE ASSOCIATED WITH RETINAL GANGLION CELL DEGENERATION INSERM (Institut National de la Santé et de la Recherche Médicale) (FR) 2011-09-22 WO claimed
WO-2010089355-A1 TAURINE OR TAURINE-LIKE SUBSTANCES FOR THE PREVENTION AND TREATMENT OF A DISEASE ASSOCIATED WITH RETINAL GANGLION CELL DEGENERATION INSERM (Institut National de la Santé et de la Recherche Médicale) (FR) 2010-08-12 WO claimed
WO-2010018418-A1 FORMULATION BASED ON MICRONIZED CLINOPTILOLITE AS THERAPEUTIC AGENT PROVIDING HIGHLY BIOAVAILABLE SILICON NOVATECH D.O.O. (HR) 2010-02-18 WO claimed
US-4485091-A HYDROGEN PEROXIDE, OIL IN WATER EMULSION QUINODERM LIMITED (GB) 1984-11-27 US claimed
EP-4539816-A1 COMPOSITIONS AND METHODS FOR AN ORAL SUPPLEMENT TO ORAL MINOXIDIL FOR THE TREATMENT OF ALOPECIA Follea International (US) 2025-04-23 EP disclosed
WO-2025048828-A1 COMPOSITIONS AND METHODS FOR AN ORAL SUPPLEMENT TO ORAL MINOXIDIL FOR THE TREATMENT OF ALOPECIA FOLLEA INTERNATIONAL (US) 2025-03-06 WO disclosed
US-4485091-A HYDROGEN PEROXIDE, OIL IN WATER EMULSION QUINODERM LIMITED (GB) 1984-11-27 US disclosed
US-4035506-A Fluorocarbon dermal protective compositions MINNESOTA MINING AND MANUFACTURING COMPANY (US) 1977-07-12 US disclosed
US-4017615-A ESPECIALLY USEFUL FOR ANTIINFLAMMATORY TOPICAL CORTICOIDS SYNTEX CORPORATION (PM) 1977-04-12 US disclosed