SCHEMBL5259083

SCHEMBL5259083

O=C(O)c1cc(C2CCCC2)cc(N2CCCCS2(=O)=O)c1F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.41
ACMSD Q8TDX5 2/20 0.40
CTSD P07339 3/20 0.33
BACE1 P56817 3/20 0.33
BACE2 Q9Y5Z0 3/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMO O15229 1/20 0.32
STAT3 P40763 4/20 0.32
CALCA P06881 2/20 0.31
PARP1 P09874 1/20 0.31
ALOX5AP P20292 2/20 0.31
FEN1 P39748 2/20 0.31
PRKAB2 O43741 1/20 0.31
PRKAG1 P54619 1/20 0.31
PRKAA2 P54646 1/20 0.31
PRKAA1 Q13131 1/20 0.31
PRKAG3 Q9UGI9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5259082 0.88 ACMSD (0.40) POLBACMSDKMOSTAT3
SCHEMBL5219461 0.86 CTSD (0.36) POLBCTSDBACE1BACE2CYP3A4
SCHEMBL5219217 0.77 CTSD (0.35) POLBCTSDBACE1BACE2CYP3A4
SCHEMBL5218901 0.75 BACE1 (0.40) POLBCTSDBACE1BACE2CYP3A4
SCHEMBL5221196 0.75 CTSD (0.42) POLBCTSDBACE1BACE2CYP3A4
SCHEMBL5219458 0.75 OPRK1 (0.34) STAT3
SCHEMBL5220634 0.74 BACE1 (0.52) POLBCTSDBACE1BACE2CYP3A4
SCHEMBL5222292 0.74 POLB (0.59) POLBCTSDBACE1BACE2KMO
SCHEMBL5222900 0.71 CTSD (0.37) POLBCTSDBACE1BACE2CYP3A4
SCHEMBL5218765 0.71 CTSD (0.34) POLBCTSDBACE1BACE2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1567488-B1 HYDROXYETHYLAMINE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE GLAXO GROUP LTD (GB) 2007-02-21 EP disclosed