SCHEMBL5259145

SCHEMBL5259145

Cc1cc(C)n(-c2cccc(C(=O)NCC(c3ccc(Cl)cc3)C(C)c3ccc(Cl)cc3)c2)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
HPGD P15428 3/20 0.45
TP53 P04637 2/20 0.45
KAT6A Q92794 1/20 0.45
MAPT P10636 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
GAA P10253 2/20 0.43
LMNA P02545 1/20 0.43
ALPG P10696 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
DGAT2 Q96PD7 1/20 0.42
CYP24A1 Q07973 1/20 0.41
HSD17B10 Q99714 1/20 0.40
POLB P06746 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
NPY5R Q15761 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6325790 0.81 CNR1 (0.52) ALDH1A1HPGDTP53KAT6AMAPT
SCHEMBL5264039 0.80 KMT2A (0.53) ALDH1A1HPGDTP53MAPTKMT2A
SCHEMBL5262774 0.76 SLC6A9 (0.54) TP53KMT2AMEN1GAAHSD17B10
SCHEMBL5263063 0.76 RAB9A (0.65) ALDH1A1HPGDMAPTL3MBTL1KMT2A
SCHEMBL5260346 0.76 RAB9A (0.46) TP53KMT2AMEN1GAALMNA
SCHEMBL4693461 0.75 RAB9A (0.56) ALDH1A1HPGDMAPTKMT2AMEN1
SCHEMBL5266049 0.74 RAB9A (0.60) ALDH1A1HPGDTP53MAPTL3MBTL1
SCHEMBL4693990 0.73 POLB (0.60) HPGDKMT2AMEN1GAALMNA
SCHEMBL5265150 0.72 NOTUM (0.50) TP53MAPTKMT2AMEN1CYP24A1
SCHEMBL5262488 0.72 SLC6A9 (0.55) KMT2AMEN1CYP24A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1494997-A4 SUBSTITUTED ARYL AMIDES MERCK & CO INC (US) 2007-04-11 EP claimed
JP-2005527586-A 2005-09-15 JP claimed
EP-1494997-A1 SUBSTITUTED ARYL AMIDES Merck & Co., Inc. (US) 2005-01-12 EP claimed
WO-2003087037-A1 SUBSTITUTED ARYL AMIDES MERCK & CO., INC. (US) 2003-10-23 WO claimed
EP-1494997-A4 SUBSTITUTED ARYL AMIDES MERCK & CO INC (US) 2007-04-11 EP disclosed
EP-1494997-A1 SUBSTITUTED ARYL AMIDES Merck & Co., Inc. (US) 2005-01-12 EP disclosed
WO-2003087037-A1 SUBSTITUTED ARYL AMIDES MERCK & CO., INC. (US) 2003-10-23 WO disclosed