SCHEMBL5263063

SCHEMBL5263063

CC(c1ccc(Cl)cc1)C(CNC(=O)c1cccc(N2CCCC2=O)c1)c1ccc(Cl)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 7/20 0.65
NPC1 O15118 6/20 0.65
KMT2A Q03164 4/20 0.57
MEN1 O00255 3/20 0.57
ALDH1A1 P00352 4/20 0.54
L3MBTL1 Q9Y468 2/20 0.54
HPGD P15428 2/20 0.54
USP2 O75604 1/20 0.54
LMNA P02545 1/20 0.54
SMN1; SMN2 Q16637 3/20 0.52
TSHR P16473 2/20 0.52
GFER P55789 2/20 0.52
MAPT P10636 2/20 0.52
GAA P10253 1/20 0.52
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
POLB P06746 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5263349 0.88 MAPT (0.65) RAB9ANPC1KMT2AMEN1ALDH1A1
SCHEMBL5260346 0.85 RAB9A (0.46) RAB9ANPC1KMT2AMEN1LMNA
SCHEMBL6327703 0.81 RAB9A (0.63) RAB9ANPC1KMT2AMEN1ALDH1A1
SCHEMBL3230238 0.81 NPC1 (0.80) RAB9ANPC1KMT2AMEN1ALDH1A1
SCHEMBL5264039 0.79 KMT2A (0.53) RAB9ANPC1KMT2AMEN1ALDH1A1
SCHEMBL5259145 0.76 ALDH1A1 (0.46) RAB9ANPC1KMT2AMEN1ALDH1A1
SCHEMBL5262774 0.75 SLC6A9 (0.54) RAB9ANPC1KMT2AMEN1SMN1; SMN2
SCHEMBL743304 0.74 MEN1 (1.00) RAB9ANPC1KMT2AMEN1ALDH1A1
SCHEMBL5266049 0.73 RAB9A (0.60) RAB9ANPC1KMT2AMEN1ALDH1A1
SCHEMBL5261535 0.73 TP53 (0.56) RAB9AKMT2AMEN1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1494997-A4 SUBSTITUTED ARYL AMIDES MERCK & CO INC (US) 2007-04-11 EP claimed
JP-2005527586-A 2005-09-15 JP claimed
EP-1494997-A1 SUBSTITUTED ARYL AMIDES Merck & Co., Inc. (US) 2005-01-12 EP claimed
WO-2003087037-A1 SUBSTITUTED ARYL AMIDES MERCK & CO., INC. (US) 2003-10-23 WO claimed